SCHEMBL11028018

SCHEMBL11028018

CCOC(=O)Nc1ccc(C(O)CNC(C)C)cc1C#N

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.57
ADRB2 P07550 5/20 0.57
TSHR P16473 5/20 0.57
ADRB1 P08588 4/20 0.57
MAPK1 P28482 4/20 0.57
ADRB3 P13945 4/20 0.57
CYP3A4 P08684 3/20 0.57
NLRP3 Q96P20 1/20 0.46
CYP2C19 P33261 2/20 0.44
CYP2C9 P11712 1/20 0.44
MAPT P10636 5/20 0.43
KDM4E B2RXH2 4/20 0.43
TDP1 Q9NUW8 4/20 0.43
HSD17B10 Q99714 3/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
HIF1A Q16665 3/20 0.43
MTOR P42345 2/20 0.43
LMNA P02545 2/20 0.43
NFKB1 P19838 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11431747 0.99 ADRB2 (0.56) CYP1A2ADRB2TSHRADRB1MAPK1
SCHEMBL11027641 0.86 NLRP3 (0.46) CYP1A2ADRB2TSHRADRB1MAPK1
SCHEMBL16794796 0.83 NLRP3 (0.52) CYP1A2NLRP3CYP2C19CYP2C9KDM4E
SCHEMBL4430153 0.81 ADRB3 (0.59) CYP1A2ADRB2TSHRADRB1MAPK1
SCHEMBL10659631 0.80 TSHR (0.69) CYP1A2ADRB2TSHRADRB1MAPK1
SCHEMBL404869 0.78 CYP1A2 (0.67) CYP1A2TSHRNLRP3CYP2C19CYP2C9
SCHEMBL10711662 0.76 NLRP3 (0.56) CYP1A2NLRP3CYP2C19CYP2C9KDM4E
SCHEMBL5972201 0.76 NLRP3 (0.56) CYP1A2MAPK1NLRP3CYP2C19CYP2C9
SCHEMBL27729156 0.75 NLRP3 (0.46) CYP1A2NLRP3CYP2C19CYP2C9KDM4E
SCHEMBL22988070 0.74 NLRP3 (0.55) CYP1A2MAPK1CYP3A4NLRP3CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0057900-B1 ANIMAL FEED ADDITIVE FOR IMPROVING GROWTH Dr. Karl Thomae GmbH (DE) 1985-05-08 EP claimed
US-4214001-A ANALGESICS, ANTISPASMODICS AND ANTIASTHMATICS BOEHRINGER INGELHEIM GMBH (DE) 1980-07-22 US claimed
EP-0057900-B1 ANIMAL FEED ADDITIVE FOR IMPROVING GROWTH Dr. Karl Thomae GmbH (DE) 1985-05-08 EP disclosed
EP-0057900-A1 Animal feed additive for improving growth Dr. Karl Thomae GmbH (DE) 1982-08-18 EP disclosed
EP-0057900-A1 Animal feed additive for improving growth Dr. Karl Thomae GmbH (DE) 1982-08-18 EP disclosed
EP-0008715-B1 PHENYLETHANOLAMINES FOR USE IN COMBATTING INFLAMMATORY CONDITIONS Dr. Karl Thomae GmbH (DE) 1981-11-25 EP disclosed
US-4244967-A ANTIIFLAMMATORY AND ANTIRHEUMATIC PROPERTIES BOEHRINGER INGELHEIM GMBH (DE) 1981-01-13 US disclosed
US-4214001-A ANALGESICS, ANTISPASMODICS AND ANTIASTHMATICS BOEHRINGER INGELHEIM GMBH (DE) 1980-07-22 US disclosed
EP-0008715-A1 Phenylethanolamines for use in combatting inflammatory conditions Dr. Karl Thomae GmbH (DE) 1980-03-19 EP disclosed