SCHEMBL11032765

SCHEMBL11032765

O=C1COc2c(C(=O)CBr)ccc(OCc3ccccc3)c2N1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.39
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.37
ADRB2 P07550 2/20 0.37
DRD2 P14416 1/20 0.37
DRD1 P21728 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
POLB P06746 2/20 0.36
ADRB1 P08588 2/20 0.36
HPGDS O60760 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9909633 0.89 SMN1; SMN2 (0.44) FOLH1BRD4CREBBPL3MBTL1MAPT
SCHEMBL1559916 0.89 ADRB2 (0.39) FOLH1BRD4CREBBPL3MBTL1MAPT
SCHEMBL1558720 0.87 MAPT (0.50) FOLH1BRD4CREBBPL3MBTL1MAPT
Water SCHEMBL6406913 0.85 ADRB2 (0.39) FOLH1BRD4CREBBPL3MBTL1MAPT
SCHEMBL632293 0.85 ADRB1 (0.40) FOLH1BRD4CREBBPL3MBTL1MAPT
SCHEMBL13437541 0.84 BRD4 (0.35) FOLH1BRD4CREBBPL3MBTL1MAPT
SCHEMBL10982611 0.83 BRD4 (0.37) FOLH1BRD4CREBBPL3MBTL1MAPT
Hydrochloric Acid SCHEMBL11216398 0.81 ADRB2 (0.35) BRD4CREBBPL3MBTL1MAPTCYP2C9
SCHEMBL632130 0.80 ADRB2 (0.37) BRD4CREBBPL3MBTL1MAPTCYP2C9
SCHEMBL1764304 0.77 MAOA (0.46) CREBBPMAPTSMN1; SMN2ADRB2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0073505-B1 BENZO-HETEROCYCLES BOEHRINGER INGELHEIM KG (DE) 1985-11-27 EP disclosed
US-4460581-A ANTISPASMODIC AGENTS, ANTIALLERGENS BOEHRINGER INGELHEIM KG (DE) 1984-07-17 US disclosed
EP-0073505-A1 Benzo-heterocycles BOEHRINGER INGELHEIM KG (DE) 1983-03-09 EP disclosed