SCHEMBL11034153

SCHEMBL11034153

Fc1cccc(C2=CCCCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CASP3 P42574 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
ACMSD Q8TDX5 2/20 0.44
TAAR1 Q96RJ0 3/20 0.42
ESR2 Q92731 1/20 0.40
SERPINE1 P05121 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
PSMB5 P28074 2/20 0.38
GALR1 P47211 1/20 0.38
FFAR2 O15552 1/20 0.38
HTR1A P08908 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
NISCH Q9Y2I1 1/20 0.38
PRMT5 O14744 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1255411 0.98 CHRNB4 (0.47) CHRNB4CHRNA3CASP3SENP8SENP7
SCHEMBL9377901 0.84 CHRNB4 (0.46) CHRNB4CHRNA3TAAR1ESR2GALR1
SCHEMBL1257281 0.82 CASP3 (0.47) CHRNB4CHRNA3CASP3SENP8SENP7
SCHEMBL17070223 0.80 CASP3 (0.46) CHRNB4CHRNA3CASP3SENP8SENP7
SCHEMBL3243443 0.78 CASP3 (0.47) CASP3SENP8SENP7SENP6ACMSD
SCHEMBL28039116 0.78 CHRNB4 (0.56) CHRNB4CHRNA3TAAR1ESR2GALR1
SCHEMBL971143 0.78 CHRNB4 (0.49) CHRNB4CHRNA3ACMSDSERPINE1TDP1
SCHEMBL18905371 0.78 ACMSD (0.44) CASP3SENP8SENP7SENP6ACMSD
SCHEMBL19910204 0.78 CHRNB4 (0.49) CHRNB4CHRNA3ACMSDSERPINE1TDP1
SCHEMBL417070 0.78 ACMSD (0.51) CHRNB4CHRNA3ACMSDESR2SERPINE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4255429-A1 3-HETEROARYL PYRROLIDINE AND PIPERIDINE OREXIN RECEPTOR AGONISTS Merck Sharp & Dohme LLC (US) 2023-10-11 EP claimed
WO-2022119888-A1 3-HETEROARYL PYRROLIDINE AND PIPERIDINE OREXIN RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2022-06-09 WO claimed
JP-59042328-A None JP disclosed
WO-2020120606-A1 NEW PYRROLIDINE-2-CARBOXYLIC ACID DERIVATIVES FOR TREATING PAIN AND PAIN RELATED CONDITIONS ESTEVE PHARMACEUTICALS, S.A. (ES) 2020-06-18 WO disclosed
JP-S5942328-A 3-FLUOROPHENYLCYCLOHEXENE DERIVATIVE CHISSO CORP 1984-03-08 JP disclosed