SCHEMBL11034285

SCHEMBL11034285

C=CCSc1cccc(-c2nc3cncnc3[nH]2)c1OC

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.32
HPGD P15428 3/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
TP53 P04637 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PDE5A O76074 2/20 0.31
KDM4E B2RXH2 1/20 0.31
USP2 O75604 1/20 0.31
GAA P10253 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
FGFR1 P11362 1/20 0.30
FGFR2 P21802 1/20 0.30
PKM P14618 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11010987 0.84 KDM4E (0.39) ALDH1A1HPGDNPC1RAB9ATP53
SCHEMBL11034287 0.84 PDE5A (0.40) ALDH1A1HPGDNPC1RAB9ATP53
SCHEMBL11007618 0.84 PDE5A (0.31) ALDH1A1HPGDPDE5AKDM4EUSP2
SCHEMBL11007368 0.81 FGFR1 (0.38) ALDH1A1HPGDTP53SMN1; SMN2PDE5A
SCHEMBL11007757 0.80 MAPT (0.34) ALDH1A1HPGDNPC1RAB9ATP53
SCHEMBL11010240 0.78 AMY1A (0.34) ALDH1A1HPGDNPC1RAB9ATP53
SCHEMBL11009397 0.78 PDE5A (0.35) ALDH1A1HPGDNPC1RAB9ATP53
SCHEMBL11011531 0.73 FGFR1 (0.38) ALDH1A1HPGDMEN1KMT2APDE5A
SCHEMBL11005174 0.73 PDE5A (0.32) ALDH1A1PDE5AFGFR1FGFR2TSHR
SCHEMBL11011418 0.73 PDE5A (0.32) ALDH1A1PDE5AFGFR1FGFR2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142075-A2 Purine derivatives, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-05-22 EP disclosed