SCHEMBL11038201

SCHEMBL11038201

CCCOC(=O)Cc1ccc(N)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.47
LMNA P02545 2/20 0.47
CYP3A4 P08684 2/20 0.47
TSHR P16473 2/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
PDE4D Q08499 1/20 0.47
ALDH1A1 P00352 4/20 0.45
GAA P10253 1/20 0.45
NPC1 O15118 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45
MAOA P21397 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
PPIB P23284 1/20 0.44
PPIA P62937 1/20 0.44
PPID Q08752 1/20 0.44
PPIG Q13427 1/20 0.44
CYP19A1 P11511 1/20 0.44
YWHAG P61981 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10899541 0.90 CYP1A2 (0.61) CYP1A2LMNACYP3A4TSHRCYP2C9
SCHEMBL11146009 0.87 ALDH1A1 (0.63) CYP1A2LMNACYP3A4TSHRCYP2C9
SCHEMBL85523 0.85 PPID (0.58) CYP1A2LMNACYP3A4TSHRALDH1A1
SCHEMBL13826445 0.84 ALDH1A1 (0.48) CYP3A4TSHRCYP2C19ALDH1A1GAA
SCHEMBL1885468 0.84 ALDH1A1 (0.58) CYP1A2LMNATSHRCYP2C19ALDH1A1
SCHEMBL5542953 0.84 ALDH1A1 (0.46) CYP1A2LMNATSHRALDH1A1GAA
SCHEMBL2400474 0.84 KMT2A (0.51) CYP1A2TSHRCYP2C9ALDH1A1GAA
Hydrochloric Acid SCHEMBL77910 0.84 PPIB (0.56) CYP1A2LMNACYP3A4TSHRALDH1A1
SCHEMBL28010049 0.83 TDP1 (0.56) CYP1A2LMNACYP3A4TSHRCYP2C9
SCHEMBL13481189 0.82 KLK7 (0.52) ALDH1A1GAAMAPTRAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117417285-B Isomanka key intermediate and preparation method thereof 苏中药业集团股份有限公司 2025-04-25 CN disclosed
CN-117417285-A Isomanka key intermediate and preparation method thereof 苏中药业集团股份有限公司 2024-01-19 CN disclosed
US-9073905-B2 Rock inhibitors AMAKEM NV (BE) 2015-07-07 US disclosed
US-9073905-B2 Rock inhibitors AMAKEM NV (BE) 2015-07-07 US disclosed
WO-2015060359-A1 NOVEL DIAMINE, POLYAMIC ACID, AND POLYIMIDE 日産化学工業株式会社 2015-04-30 WO disclosed
US-20140057942-A1 NOVEL ROCK INHIBITORS AMAKEM NV (BE) 2014-02-27 US disclosed
US-20140057942-A1 NOVEL ROCK INHIBITORS AMAKEM NV (BE) 2014-02-27 US disclosed
WO-2012146724-A2 NOVEL ROCK INHIBITORS AMAKEM NV (BE) 2012-11-01 WO disclosed
EP-0052296-B1 GLUTAMINE DERIVATIVES USABLE FOR CURING IMMUNE DISEASES, METHODS FOR THEIR PREPARATION AND COMPOSITIONS COMPRISING SAID DERIVATIVES MITSUBISHI KASEI CORPORATION (JP) 1984-06-27 EP disclosed
US-4439448-A IMMUNOMODULATING ACTIVITY MITSUBISHI CHEMICAL INDUSTRIES LTD. (JP) 1984-03-27 US disclosed
EP-0052296-A1 Glutamine derivatives usable for curing immune diseases, methods for their preparation and compositions comprising said derivatives MITSUBISHI KASEI CORPORATION (JP) 1982-05-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140057942-A1 NOVEL ROCK INHIBITORS ROCK1, ROCK2, CIT CYP1A2 636/4885LMNA 3808/4885CYP3A4 1301/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.