SCHEMBL11038671

SCHEMBL11038671

CCOc1cc2c(cc1OCC)CC(=O)[N]C=C2

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.40
BRD4 O60885 1/20 0.36
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
TP53 P04637 2/20 0.33
MDM2 Q00987 2/20 0.33
PDE4D Q08499 2/20 0.33
TSHR P16473 3/20 0.33
CYP3A4 P08684 1/20 0.33
POLB P06746 2/20 0.31
LMNA P02545 2/20 0.31
MAPT P10636 1/20 0.31
S1PR1 P21453 1/20 0.31
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1533850 0.83 BRD4 (0.53) ACHEBRD4KDM4EALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL11040765 0.75 TSHR (0.36) ACHEKDM4EALDH1A1PDE4DTSHR
SCHEMBL11043204 0.75 BRD4 (0.44) BRD4KDM4EALDH1A1CYP3A4LMNA
SCHEMBL11041593 0.73 GAA (0.51) ACHEBRD4KDM4EALDH1A1TP53
SCHEMBL11057303 0.71 MAPT (0.40) BRD4KDM4EALDH1A1PDE4DTSHR
SCHEMBL11040367 0.71 MAPT (0.40) BRD4KDM4EALDH1A1PDE4DTSHR
Hydrochloric Acid SCHEMBL11059748 0.71 MAPT (0.42) BRD4KDM4EALDH1A1PDE4DTSHR
Hydrochloric Acid SCHEMBL11051850 0.71 MAPT (0.42) BRD4KDM4EALDH1A1PDE4DTSHR
SCHEMBL11039717 0.69 BRD4 (0.41) BRD4KDM4EALDH1A1PDE4DTSHR
SCHEMBL24465258 0.68 MAPT (0.52) ACHEKDM4EALDH1A1TP53MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116444-A2 Improvements in or relating to benzazepine derivatives ELI LILLY AND COMPANY (US) 1984-08-22 EP disclosed