SCHEMBL11041593

SCHEMBL11041593

CCOc1cc2c(cc1OCC)CC(=O)NC=C2

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.51
ACHE P22303 2/20 0.40
BRD4 O60885 1/20 0.36
S1PR1 P21453 1/20 0.35
PDE4A P27815 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.33
MDM2 Q00987 1/20 0.33
PDE4D Q08499 2/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.32
MAPT P10636 2/20 0.32
ABCC4 O15439 1/20 0.32
ABCB11 O95342 1/20 0.32
CHRM2 P08172 1/20 0.32
ADRA2A P08913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL333847 0.83 GAA (0.63) GAAACHEBRD4KDM4EALDH1A1
SCHEMBL11038245 0.78 GAA (0.53) GAA
SCHEMBL11041605 0.77 BRD4 (0.39) GAABRD4KDM4EALDH1A1PDE4D
Oxalic Acid SCHEMBL15319252 0.77 GAA (0.56) GAABRD4MAPK1CYP3A4KMT2A
SCHEMBL28634068 0.76 GAA (0.58) GAABRD4MAPK1CYP3A4KMT2A
SCHEMBL15906664 0.75 GAA (0.57) GAAACHEBRD4ALDH1A1
SCHEMBL11045652 0.75 GAA (0.57) GAABRD4KDM4EALDH1A1MAPK1
SCHEMBL13593675 0.74 GAA (0.53) GAABRD4PDE4APDE4DMAPK1
SCHEMBL9214465 0.74 GAA (0.55) GAAHTT
SCHEMBL11038671 0.73 ACHE (0.40) ACHEBRD4S1PR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116444-A2 Improvements in or relating to benzazepine derivatives ELI LILLY AND COMPANY (US) 1984-08-22 EP disclosed