SCHEMBL11039262

SCHEMBL11039262

COC(=O)c1ccc(CC(C)NCC(O)c2cccc(C(F)(F)F)c2)cc1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 11/20 0.49
ADRA1A P35348 3/20 0.49
USP2 O75604 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 2/20 0.49
ADRA2C P18825 2/20 0.49
HTR2A P28223 2/20 0.49
SLC6A4 P31645 2/20 0.49
DRD3 P35462 2/20 0.49
HTR2B P41595 2/20 0.49
NR1I2 O75469 1/20 0.49
HTR1A P08908 1/20 0.49
ADRA2A P08913 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
ADRA2B P18089 1/20 0.49
CHRM3 P20309 1/20 0.49
SLC6A2 P23975 1/20 0.49
HTR2C P28335 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11053844 0.89 ADRB3 (0.56) ADRB1ADRA1AUSP2CYP3A4CYP1A2
SCHEMBL9007073 0.89 ADRB3 (0.56) ADRB1ADRA1AUSP2CYP3A4CYP1A2
SCHEMBL9007077 0.89 ADRB3 (0.56) ADRB1ADRA1AUSP2CYP3A4CYP1A2
Hydrochloric Acid SCHEMBL11040417 0.88 ADRB3 (0.55) ADRB1ADRA1AUSP2CYP3A4CYP1A2
SCHEMBL10773274 0.84 ADRB1 (0.60) ADRB1ADRA1AUSP2CYP3A4CYP1A2
SCHEMBL10937612 0.83 ADRB3 (0.57) ADRB1ADRA1AUSP2CYP3A4CYP1A2
SCHEMBL10772579 0.82 ADRB1 (0.69) ADRB1ADRA1AUSP2CYP3A4CYP1A2
SCHEMBL9006832 0.82 ADRB1 (0.69) ADRB1ADRA1AUSP2CYP3A4CYP1A2
SCHEMBL9007030 0.82 ADRB1 (0.69) ADRB1ADRA1AUSP2CYP3A4CYP1A2
SCHEMBL10890320 0.81 SLC2A1 (0.56) ADRB1ADRA1ACYP3A4CYP2D6ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0040915-B1 ARYLETHANOLAMINE DERIVATIVES, THEIR PREPARATION AND USE IN PHARMACEUTICAL COMPOSITIONS BEECHAM GROUP PLC (GB) 1984-03-21 EP disclosed
US-4385066-A DIETETICS, HYPERGLYCEMIC AGENTS ANTIINFLAMMATORY AGENTS BEECHAM GROUP LIMITED (GB) 1983-05-24 US disclosed
EP-0040915-A1 Arylethanolamine derivatives, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-12-02 EP disclosed