SCHEMBL11040653

SCHEMBL11040653

COc1c(C)cc(Cl)cc1C1OC(=O)NC1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.49
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LRRK2 Q5S007 1/20 0.33
POLB P06746 1/20 0.33
BRD4 O60885 3/20 0.32
PKM P14618 1/20 0.32
CES1 P23141 1/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
CYP19A1 P11511 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11040514 0.80 CA2 (0.48) CA2ALDH1A1KDM4ETSHRSMN1; SMN2
SCHEMBL11040511 0.76 CA2 (0.60) CA2ALDH1A1TSHR
SCHEMBL11040852 0.76 CA2 (0.50) CA2BRD4GRIN2DGRIN3BGRIN1
SCHEMBL11040233 0.75 CA2 (0.59) CA2ALDH1A1TSHR
SCHEMBL11040237 0.75 CA2 (0.59) CA2ALDH1A1TSHR
SCHEMBL10546613 0.74 CA2 (0.48) CA2TSHRSMN1; SMN2GRIN2DGRIN3B
SCHEMBL10927277 0.73 ALDH1A1 (0.47) ALDH1A1KDM4ETSHRSMN1; SMN2LRRK2
SCHEMBL10499858 0.72 ALDH1A1 (0.39) CA2ALDH1A1KDM4ETSHRSMN1; SMN2
SCHEMBL11043516 0.69 CA2 (0.62) CA2ALDH1A1TSHRSMN1; SMN2KMT2A
SCHEMBL11040416 0.68 HTR2C (0.48) CA2TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4448971-A Hypoglycemic 5-phenyl-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1984-05-15 US disclosed
US-4407811-A Hypoglycemic 5-substituted oxazolidine-2,4-diones PFIZER INC. (US) 1983-10-04 US disclosed
US-4399296-A TRIMETHYLSILYL CYANOHYDRIN INTERMEDIATES PFIZER INC. (US) 1983-08-16 US disclosed
US-4367234-A HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1983-01-04 US disclosed