SCHEMBL11040907

SCHEMBL11040907

Clc1ccc2c(cnn2Cc2cccc(NC3=NCCN3)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
ADRA2A P08913 9/20 0.43
ADRA2B P18089 5/20 0.43
ADRA2C P18825 5/20 0.43
PTGIR P43119 1/20 0.42
MEN1 O00255 1/20 0.41
SLC22A1 O15245 1/20 0.41
SLC22A3 O75751 1/20 0.41
LMNA P02545 1/20 0.41
HTR1A P08908 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
HRH2 P25021 1/20 0.41
ADRA1D P25100 1/20 0.41
CYP2C19 P33261 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
OPRK1 P41145 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11043668 0.88 PTGIR (0.50) ADRA2AADRA2BADRA2CPTGIRADRA1D
SCHEMBL11045568 0.87 ERBB2 (0.51) EGFRERBB2ADRA2AADRA2BADRA2C
SCHEMBL11762296 0.75 ADRA2A (0.59) ADRA2AADRA2BADRA2CPTGIRMEN1
SCHEMBL9917342 0.72 KMO (0.57) EGFRERBB2
SCHEMBL11042229 0.72 ADRA2A (0.46) ADRA2AADRA2BADRA2CMEN1SLC22A1
SCHEMBL11046783 0.72 ADRA2A (0.47) ADRA2AADRA2BADRA2CPTGIRMEN1
SCHEMBL11047792 0.72 ADRA2A (0.52) ADRA2AADRA2BADRA2CPTGIRMEN1
SCHEMBL14367989 0.72 NISCH (0.58) ADRA2AADRA2BADRA2CPTGIRADRA1D
SCHEMBL11045827 0.70 ADRA2A (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL11039489 0.70 LMNA (0.51) ADRA2AADRA2BADRA2CMEN1SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4436913-A HYPOTENSIVE AGENTS SIEGFRIED AKTIENGESELLSCHAFT (CH) 1984-03-13 US claimed
EP-0047328-B1 1H AND 2H INDAZOLE DERIVATIVES AND MEDICAMENT CONTAINING THEM SIEGFRIED AKTIENGESELLSCHAFT (CH) 1984-05-09 EP disclosed