SCHEMBL11041342

SCHEMBL11041342

C=CCc1nc2c(c(=O)n(O)c(=O)n2O)n1CCCCC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 8/20 0.45
SMN1; SMN2 Q16637 5/20 0.45
HTT P42858 4/20 0.45
LMNA P02545 3/20 0.45
MAPK1 P28482 3/20 0.45
GALR3 O60755 1/20 0.45
RAB9A P51151 1/20 0.45
ALDH1A1 P00352 7/20 0.43
HSD17B10 Q99714 5/20 0.43
RECQL P46063 2/20 0.43
TP53 P04637 2/20 0.43
L3MBTL1 Q9Y468 3/20 0.42
GAA P10253 1/20 0.42
CNOT7 Q9UIV1 4/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
GLA P06280 1/20 0.40
USP2 O75604 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11041337 0.85 HTT (0.42) TSHRSMN1; SMN2HTTLMNAMAPK1
SCHEMBL11044975 0.82 USP2 (0.41) SMN1; SMN2HTTLMNAMAPK1ALDH1A1
SCHEMBL11498915 0.69 TSHR (0.59) TSHRSMN1; SMN2LMNAMAPK1ALDH1A1
SCHEMBL11044972 0.69 ADORA2B (0.42) HTTLMNAALDH1A1HSD17B10L3MBTL1
SCHEMBL5272641 0.67 USP2 (0.51) TSHRSMN1; SMN2HTTLMNAMAPK1
SCHEMBL19407022 0.64 TSHR (0.56) TSHRSMN1; SMN2HTTLMNAMAPK1
SCHEMBL3188422 0.64 CYP1A2 (0.62) TSHRSMN1; SMN2HTTLMNAMAPK1
SCHEMBL13247924 0.63 CYP1A2 (0.58) TSHRSMN1; SMN2HTTLMNAMAPK1
SCHEMBL3169929 0.63 USP2 (0.52) TSHRSMN1; SMN2HTTLMNAMAPK1
SCHEMBL6102280 0.62 USP2 (0.51) TSHRSMN1; SMN2HTTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0075850-B1 PHARMACEUTICAL PREPARATIONS CONTAINING VICINAL DIHYDROXYALKYL XANTHINES, PROCESS FOR THE PREPARATION OF THE XANTHINES AND THE APPROPRIATE INTERMEDIATES THEREFOR HOECHST AKTIENGESELLSCHAFT (DE) 1985-12-18 EP claimed