SCHEMBL11044975

SCHEMBL11044975

C=CCc1nc2c(c(=O)n(O)c(=O)n2O)n1CC=C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.41
LMNA P02545 4/20 0.38
HTT P42858 3/20 0.38
CYP3A4 P08684 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
ALDH1A1 P00352 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ADORA2B P29275 4/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
POLB P06746 1/20 0.34
ADORA2A P29274 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
HPGD P15428 1/20 0.33
BLM P54132 1/20 0.33
HSD17B10 Q99714 1/20 0.33
RCE1 Q9Y256 1/20 0.33
NCOA1 Q15788 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11044972 0.83 ADORA2B (0.42) USP2LMNAHTTCYP3A4L3MBTL1
SCHEMBL11041342 0.82 TSHR (0.45) USP2LMNAHTTCYP3A4L3MBTL1
SCHEMBL11041337 0.69 HTT (0.42) LMNAHTTL3MBTL1ALDH1A1NPSR1
SCHEMBL11668144 0.69 ADORA2B (0.45) USP2LMNAHTTCYP3A4ALDH1A1
SCHEMBL2948020 0.68 ADORA2B (0.46) USP2LMNAHTTL3MBTL1ALDH1A1
SCHEMBL5272641 0.67 USP2 (0.51) USP2LMNAHTTL3MBTL1ALDH1A1
SCHEMBL21393356 0.66 MEN1 (0.56) USP2LMNACYP3A4ALDH1A1NPSR1
SCHEMBL10818058 0.65 ALDH1A1 (0.38) CYP3A4ALDH1A1ADORA2BMEN1KMT2A
SCHEMBL1758396 0.64 CYP3A4 (0.42) USP2CYP3A4ALDH1A1NPSR1ADORA2B
SCHEMBL11029795 0.63 ADORA2B (0.46) USP2LMNAHTTCYP3A4L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0075850-B1 PHARMACEUTICAL PREPARATIONS CONTAINING VICINAL DIHYDROXYALKYL XANTHINES, PROCESS FOR THE PREPARATION OF THE XANTHINES AND THE APPROPRIATE INTERMEDIATES THEREFOR HOECHST AKTIENGESELLSCHAFT (DE) 1985-12-18 EP claimed