SCHEMBL11041337

SCHEMBL11041337

C=CCc1nc2c(c(=O)n(CCCCC)c(=O)n2O)n1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.42
MAPK1 P28482 2/20 0.42
LMNA P02545 2/20 0.42
TSHR P16473 2/20 0.42
GALR3 O60755 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 4/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TNF P01375 1/20 0.39
CNOT7 Q9UIV1 4/20 0.39
ALDH1A1 P00352 2/20 0.39
RECQL P46063 1/20 0.39
PDE4A P27815 3/20 0.39
PDE4B Q07343 3/20 0.39
PDE4C Q08493 3/20 0.39
PDE4D Q08499 3/20 0.39
ADORA2A P29274 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11041342 0.85 TSHR (0.45) HTTMAPK1LMNATSHRGALR3
SCHEMBL11044972 0.82 ADORA2B (0.42) HTTLMNAHSD17B10L3MBTL1MEN1
SCHEMBL5272641 0.75 USP2 (0.51) HTTMAPK1LMNATSHRGALR3
SCHEMBL11044975 0.69 USP2 (0.41) HTTMAPK1LMNASMN1; SMN2HSD17B10
SCHEMBL11033010 0.67 ADORA2B (0.48) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11498915 0.67 TSHR (0.59) MAPK1LMNATSHRSMN1; SMN2HSD17B10
SCHEMBL13247924 0.66 CYP1A2 (0.58) HTTMAPK1LMNATSHRGALR3
SCHEMBL19407022 0.64 TSHR (0.56) HTTMAPK1LMNATSHRGALR3
SCHEMBL3115778 0.64 CYP1A2 (0.52) HTTMAPK1LMNATSHRGALR3
SCHEMBL11466640 0.64 PDE4A (0.65) LMNAMEN1KMT2ACNOT7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0075850-B1 PHARMACEUTICAL PREPARATIONS CONTAINING VICINAL DIHYDROXYALKYL XANTHINES, PROCESS FOR THE PREPARATION OF THE XANTHINES AND THE APPROPRIATE INTERMEDIATES THEREFOR HOECHST AKTIENGESELLSCHAFT (DE) 1985-12-18 EP claimed