SCHEMBL11041566

SCHEMBL11041566

O=C(Nc1ccc(Cl)cc1)ONC1=Nc2ccc(Br)cc2C(c2ccccc2F)=NC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
AURKA O14965 1/20 0.37
TP53 P04637 1/20 0.37
CHRM1 P11229 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CCKBR P32239 1/20 0.36
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11053089 0.94 LMNA (0.44) LMNAALDH1A1AURKATP53CHRM1
SCHEMBL11168627 0.92 MEN1 (0.42) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11046042 0.91 TP53 (0.43) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11169424 0.91 GABRA1 (0.40) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11044126 0.91 CYP1A2 (0.37) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11170761 0.91 CYP1A2 (0.43) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11057804 0.91 LMNA (0.44) LMNAAURKATP53CHRM1CYP3A4
SCHEMBL11166541 0.89 GABRA1 (0.42) GABRA1GABRA5GABRA3GABRA2GABRB2
SCHEMBL11039376 0.88 TP53 (0.46) LMNAALDH1A1NPC1RAB9AKMT2A
SCHEMBL11166336 0.88 CYP1A2 (0.41) GABRA1GABRA5GABRA3GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0041242-B1 CARBAMOYLOXYAMINO-1,4-BENZODIAZEPINES, THEIR PREPARATION AND MEDICINES CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1984-07-11 EP disclosed
US-4395409-A ANXIOLYTIC AGENT HOECHST AKTIENGESELLSCHAFT (DE) 1983-07-26 US disclosed