SCHEMBL11057804

SCHEMBL11057804

O=C(Nc1ccccc1)ONC1=Nc2ccc(Cl)cc2C(c2ccccc2F)=NC1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
AURKA O14965 2/20 0.43
TP53 P04637 1/20 0.42
CHRM1 P11229 1/20 0.41
CYP3A4 P08684 2/20 0.38
DRD3 P35462 2/20 0.38
OPRK1 P41145 2/20 0.38
SLC22A1 O15245 1/20 0.38
ABCB11 O95342 1/20 0.38
PDE4D Q08499 1/20 0.38
HTR1A P08908 1/20 0.37
HTR3A P46098 1/20 0.37
KCNH2 Q12809 1/20 0.37
GHSR Q92847 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11053089 0.97 LMNA (0.44) LMNAAURKATP53CHRM1CYP3A4
SCHEMBL11039376 0.95 TP53 (0.46) LMNAAURKATP53CHRM1CYP3A4
SCHEMBL11160221 0.93 TP53 (0.44) LMNAAURKATP53CHRM1CYP3A4
SCHEMBL11169123 0.92 LMNA (0.42) LMNAAURKATP53CHRM1CYP3A4
SCHEMBL11046042 0.91 TP53 (0.43) LMNAAURKATP53CHRM1
SCHEMBL11041566 0.91 GABRA1 (0.41) LMNAAURKATP53CHRM1CYP3A4
SCHEMBL11044384 0.89 TP53 (0.41) LMNAAURKATP53CHRM1CYP3A4
SCHEMBL11168627 0.88 MEN1 (0.42) LMNAAURKATP53CHRM1CYP3A4
SCHEMBL11043502 0.88 NPSR1 (0.44) TP53CHRM1OPRK1PDE4DKCNH2
SCHEMBL11171819 0.88 LMNA (0.42) LMNAAURKATP53CHRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0041242-B1 CARBAMOYLOXYAMINO-1,4-BENZODIAZEPINES, THEIR PREPARATION AND MEDICINES CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1984-07-11 EP disclosed
US-4395409-A ANXIOLYTIC AGENT HOECHST AKTIENGESELLSCHAFT (DE) 1983-07-26 US disclosed
EP-0041242-A1 Carbamoyloxyamino-1,4-benzodiazepines, their preparation and medicines containing them HOECHST AKTIENGESELLSCHAFT (DE) 1981-12-09 EP disclosed