SCHEMBL11041640

SCHEMBL11041640

COc1cc2c(cc1OC)CC(N)=NC=C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.45
CYP3A4 P08684 3/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 6/20 0.36
ALDH1A1 P00352 5/20 0.36
GLA P06280 3/20 0.36
MAOA P21397 3/20 0.36
GAA P10253 3/20 0.33
HPGD P15428 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP2C9 P11712 1/20 0.32
MAPK1 P28482 1/20 0.32
PKM P14618 1/20 0.32
RAD52 P43351 1/20 0.32
EHMT2 Q96KQ7 1/20 0.32
CHEK1 O14757 1/20 0.32
CYP2D6 P10635 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11040043 0.98 BRD4 (0.44) BRD4CYP3A4MAPTKDM4EALDH1A1
SCHEMBL11057303 0.90 MAPT (0.40) BRD4CYP3A4MAPTKDM4EALDH1A1
SCHEMBL11040367 0.90 MAPT (0.40) BRD4CYP3A4MAPTKDM4EALDH1A1
Hydrochloric Acid SCHEMBL11059748 0.89 MAPT (0.42) BRD4CYP3A4MAPTKDM4EALDH1A1
Hydrochloric Acid SCHEMBL11051850 0.89 MAPT (0.42) BRD4CYP3A4MAPTKDM4EALDH1A1
Hydrochloric Acid SCHEMBL11038881 0.88 BRD4 (0.38) BRD4CYP3A4MAPTGAA
Hydrochloric Acid SCHEMBL11042874 0.86 BRD4 (0.38) BRD4CYP3A4MAPTALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL11038894 0.86 MAOA (0.38) BRD4CYP3A4MAPTALDH1A1MAOA
Hydrochloric Acid SCHEMBL11051967 0.86 MAOA (0.40) BRD4ALDH1A1MAOACYP2D6HSD17B10
SCHEMBL11041298 0.81 BRD4 (0.46) BRD4CYP3A4MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116444-A2 Improvements in or relating to benzazepine derivatives ELI LILLY AND COMPANY (US) 1984-08-22 EP claimed
EP-0115961-A2 Process for preparing benzazepines ELI LILLY AND COMPANY (US) 1984-08-15 EP claimed
EP-0116444-A2 Improvements in or relating to benzazepine derivatives ELI LILLY AND COMPANY (US) 1984-08-22 EP disclosed
EP-0115961-A2 Process for preparing benzazepines ELI LILLY AND COMPANY (US) 1984-08-15 EP disclosed