SCHEMBL11043352

SCHEMBL11043352

COc1ccc(-c2csc(=S)n2-c2ccc(OC)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
HPGD P15428 3/20 0.44
HTT P42858 2/20 0.44
CUL4A Q13619 1/20 0.44
PTGS2 P35354 2/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
TP53 P04637 1/20 0.41
ALOX12 P18054 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
STAT3 P40763 1/20 0.41
MAPT P10636 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GSK3A P49840 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19116731 0.80 MAPT (0.45) KMT2AMEN1HPGDHTTPTGS2
SCHEMBL4616451 0.74 KMT2A (0.57) KMT2AMEN1HPGDHTTPTGS2
SCHEMBL17446097 0.74 LMNA (0.48) KMT2AMEN1HPGDHTTCA12
SCHEMBL4617244 0.71 CA12 (0.67) KMT2AMEN1HTTPTGS2CA12
SCHEMBL5672477 0.70 CA12 (0.48) PTGS2CA12CA1CA2CA9
SCHEMBL5674063 0.70 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL17446240 0.68 CYP11B1 (0.50) KMT2AMEN1HPGDHTTTP53
SCHEMBL5281877 0.67 KMT2A (0.65) KMT2AMEN1HTTPTGS2CA12
SCHEMBL5671527 0.67 PTGS2 (0.56) PTGS2CA12CA1CA2CA9
SCHEMBL23643023 0.67 GSK3A (0.53) KMT2AMEN1HPGDSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4451471-A Certain 2,4,5-tri-substituted thiazoles, pharmaceutical compositions containing same and methods of using same CIBA-GEIGY CORPORATION (US) 1984-05-29 US disclosed