SCHEMBL11044918

SCHEMBL11044918

O=[C]C=Cc1cccc(I)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 3/20 0.52
ENPP2 Q13822 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
NFE2L2 Q16236 2/20 0.34
FBP1 P09467 2/20 0.34
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CCNB1 P14635 1/20 0.32
CCND1 P24385 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
FAAH O00519 1/20 0.32
MGLL Q99685 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
HSD17B3 P37058 1/20 0.32
CYP19A1 P11511 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
LCK P06239 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11044915 1.00 APP (0.52) APPENPP2TRPV1NFE2L2FBP1
SCHEMBL698580 0.80 APP (0.72) APPNFE2L2CYP19A1MAOAMAOB
SCHEMBL698579 0.80 APP (0.72) APPNFE2L2CYP19A1MAOAMAOB
SCHEMBL11039441 0.76 HSD17B3 (0.56) HSD17B3MAOAMAOBNPSR1
SCHEMBL2319724 0.76 NFE2L2 (0.65) APPNFE2L2FBP1CYP1A2MAOA
SCHEMBL2319722 0.76 NFE2L2 (0.65) APPNFE2L2FBP1CYP1A2MAOA
SCHEMBL2348351 0.76 LCK (0.59) FBP1CCNB2CDK1CDK4CCNB1
SCHEMBL2348347 0.76 LCK (0.59) FBP1CCNB2CDK1CDK4CCNB1
SCHEMBL2345287 0.76 FBP1 (0.53) NFE2L2FBP1CYP1A2MAOAMAOB
SCHEMBL2349000 0.76 CYP1A2 (0.56) NFE2L2FBP1CYP1A2CYP2C9MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed