SCHEMBL11045198

SCHEMBL11045198

O=C1CCc2cc(C(=O)N3CCN(C(=O)c4ccc5c(c4)OCO5)CC3)ccc2N1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.61
HSD17B10 Q99714 2/20 0.61
HPGD P15428 7/20 0.59
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
CRBN Q96SW2 2/20 0.56
TSHR P16473 2/20 0.54
GAA P10253 1/20 0.54
GFER P55789 1/20 0.54
NR3C1 P04150 1/20 0.53
PGR P06401 1/20 0.53
SLC6A4 P31645 1/20 0.53
KCNH2 Q12809 1/20 0.53
PDE3B Q13370 1/20 0.53
PDE3A Q14432 1/20 0.53
NPC1 O15118 1/20 0.53
TP53 P04637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7350237 0.92 MAOB (0.55) ALDH1A1HSD17B10HPGDCYP1A2CYP3A4
SCHEMBL9124972 0.92 NR3C1 (0.66) ALDH1A1HSD17B10HPGDCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL7293032 0.90 MAOB (0.54) ALDH1A1HSD17B10HPGDCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11047745 0.89 ALDH1A1 (0.64) ALDH1A1TSHRSMN1; SMN2LMNAKMT2A
SCHEMBL11197452 0.85 ALDH1A1 (0.60) ALDH1A1HSD17B10HPGDCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11041952 0.85 DRD2 (0.65) ALDH1A1HSD17B10CRBNTSHRNR3C1
SCHEMBL11046347 0.83 NR3C1 (0.62) ALDH1A1HPGDCRBNTSHRNR3C1
SCHEMBL11045054 0.82 CRBN (0.62) ALDH1A1HPGDCRBNGAANR3C1
SCHEMBL7325238 0.82 CRBN (0.58) ALDH1A1HPGDCRBNNR3C1PGR
Iodide SCHEMBL11041065 0.82 NR3C1 (0.61) ALDH1A1HPGDCRBNTSHRNR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed