SCHEMBL11045581

SCHEMBL11045581

O=C(c1ccc2[nH]c(=O)ccc2c1)N1CCN(Cc2ccccc2)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.72
NPC1 O15118 1/20 0.70
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
LMNA P02545 2/20 0.62
TSHR P16473 2/20 0.62
SMN1; SMN2 Q16637 2/20 0.62
MAPK1 P28482 1/20 0.62
L3MBTL1 Q9Y468 1/20 0.62
ALDH1A1 P00352 3/20 0.56
KDM4E B2RXH2 1/20 0.56
PARP1 P09874 1/20 0.56
PDE3B Q13370 1/20 0.55
PDE3A Q14432 1/20 0.55
PKM P14618 2/20 0.55
HDAC6 Q9UBN7 1/20 0.54
SIGMAR1 Q99720 1/20 0.53
USP2 O75604 1/20 0.52
GAA P10253 1/20 0.52
CASP1 P29466 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11042987 0.98 MAPK14 (0.69) MAPK14NPC1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL11041741 0.89 MAPK14 (0.57) MAPK14NPC1MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL11042390 0.88 MAPK14 (0.56) MAPK14NPC1MEN1KMT2ALMNA
SCHEMBL11062358 0.87 SIGMAR1 (0.58) MAPK14NPC1MEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL11039487 0.86 SIGMAR1 (0.57) MAPK14NPC1MEN1KMT2AALDH1A1
SCHEMBL16573702 0.84 MAPK14 (1.00) MAPK14NPC1MEN1KMT2ALMNA
SCHEMBL11071009 0.82 DRD3 (0.66) MEN1KMT2APDE3BPDE3ASIGMAR1
Hydrochloric Acid SCHEMBL11041259 0.81 DRD3 (0.65) MEN1KMT2APDE3BPDE3ASIGMAR1
SCHEMBL5407412 0.81 MAPK14 (0.70) MAPK14NPC1MEN1KMT2ALMNA
SCHEMBL11067206 0.81 HRH3 (0.52) MAPK14NPC1MAPK1ALDH1A1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed