SCHEMBL11045925

SCHEMBL11045925

CC(C)(C)OC(=O)N(Cc1ccccc1)C1CN[C@H](C(=O)O)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.49
DPP8 Q6V1X1 1/20 0.45
DPP7 Q9UHL4 1/20 0.45
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
CETP P11597 1/20 0.40
CTSD P07339 1/20 0.39
AKT1 P31749 2/20 0.39
KDM1A O60341 2/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
DPP4 P27487 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11045927 1.00 HSD11B1 (0.49) HSD11B1DPP8DPP7JAK2JAK1
SCHEMBL26966078 1.00 HSD11B1 (0.49) HSD11B1DPP8DPP7JAK2JAK1
SCHEMBL30722334 1.00 HSD11B1 (0.49) HSD11B1DPP8DPP7JAK2JAK1
SCHEMBL26966058 0.89 HSD11B1 (0.39) HSD11B1DPP8DPP7JAK2JAK1
SCHEMBL30722353 0.89 HSD11B1 (0.39) HSD11B1DPP8DPP7JAK2JAK1
SCHEMBL27273561 0.84 HSD11B1 (0.48) HSD11B1DPP8DPP7JAK2JAK1
SCHEMBL6980390 0.83 CTSD (0.53) HSD11B1JAK2JAK1HDAC3HDAC1
SCHEMBL895157 0.82 HSD11B1 (0.53) HSD11B1JAK2JAK1HDAC3HDAC1
SCHEMBL26966073 0.81 CYP1A2 (0.37) HSD11B1CYP2D6
SCHEMBL10207431 0.80 HSD11B1 (0.56) HSD11B1JAK2JAK1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4462943-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1984-07-31 US disclosed
EP-0052991-A1 Carboxyalkyl amino acid derivatives of various substituted prolines E.R. Squibb & Sons, Inc. (US) 1982-06-02 EP disclosed