SCHEMBL11046359

SCHEMBL11046359

Cc1cccc(C)c1-n1cnc(CO)c1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CPB1 P15086 1/20 0.39
CPB2 Q96IY4 1/20 0.39
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
NOTUM Q6P988 8/20 0.37
HCAR1 Q9BXC0 1/20 0.36
PDE10A Q9Y233 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
GRM5 P41594 2/20 0.35
GRM1 Q13255 2/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KDM4E B2RXH2 1/20 0.35
DDX3X O00571 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052371 0.84 NOTUM (0.36) CPB1CPB2PDE3BPDE3ANOTUM
SCHEMBL11048752 0.83 CPB1 (0.43) CPB1CPB2PDE3BPDE3ANOTUM
SCHEMBL11046403 0.83 CPB1 (0.54) CPB1CPB2PDE3BPDE3ANOTUM
SCHEMBL11101125 0.81 PDE3B (0.39) CPB1CPB2PDE3BPDE3ANOTUM
SCHEMBL11051360 0.79 NOTUM (0.36) CPB1CPB2PDE3BPDE3ANOTUM
SCHEMBL14704080 0.77 CYP2E1 (0.49) PDE3BPDE3AHCAR1ALDH1A1TSHR
SCHEMBL11047728 0.77 PDE3B (0.40) CPB1CPB2PDE3BPDE3ANOTUM
SCHEMBL4432563 0.75 NOTUM (0.51) CPB1CPB2PDE3BPDE3ANOTUM
SCHEMBL4427890 0.75 NOTUM (0.55) CPB2PDE3BPDE3ANOTUMHCAR1
SCHEMBL4433834 0.74 CPB2 (0.50) CPB1CPB2PDE3BPDE3ANOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0024829-B1 4-BENZYL- AND 4-BENZOYLIMIDAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME Farmos-Yhtyma Oy (FI) 1984-04-25 EP claimed
US-4443466-A DIURETICS, SEDATIVES, ANALGESICS Farmos-Yhtyma OY (Farmos Group Ltd.) (FI) 1984-04-17 US claimed
EP-0024829-A1 4-Benzyl- and 4-benzoylimidazole derivatives, processes for their preparation and pharmaceutical compositions comprising the same Farmos-Yhtyma Oy (FI) 1981-03-11 EP claimed
EP-0024829-B1 4-BENZYL- AND 4-BENZOYLIMIDAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME Farmos-Yhtyma Oy (FI) 1984-04-25 EP disclosed
US-4443466-A DIURETICS, SEDATIVES, ANALGESICS Farmos-Yhtyma OY (Farmos Group Ltd.) (FI) 1984-04-17 US disclosed
EP-0024829-A1 4-Benzyl- and 4-benzoylimidazole derivatives, processes for their preparation and pharmaceutical compositions comprising the same Farmos-Yhtyma Oy (FI) 1981-03-11 EP disclosed