SCHEMBL11047003

SCHEMBL11047003

O=C(CCC1SCCCS1)COCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.44
NPC1 O15118 1/20 0.40
GRM5 P41594 5/20 0.39
TSHR P16473 1/20 0.37
PREP P48147 1/20 0.37
CSNK1D P48730 1/20 0.36
SLC1A3 P43003 2/20 0.35
SLC1A2 P43004 2/20 0.35
SLC1A1 P43005 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 1/20 0.35
NAMPT P43490 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11601433 0.79 EPHX2 (0.48) FAAH
SCHEMBL8117531 0.78 KLK7 (0.47) NPC1GRM5MEN1KMT2A
SCHEMBL8715142 0.75 SLC1A3 (0.39) FAAHNPC1GRM5TSHRPREP
SCHEMBL24965972 0.75 TSHR (0.48) FAAHNPC1TSHR
SCHEMBL476827 0.74 TSHR (0.61) NPC1GRM5TSHRSLC1A1KMT2A
SCHEMBL8107320 0.73 SIGMAR1 (0.44) FAAHNPC1MEN1KMT2A
SCHEMBL5238071 0.73 KEAP1 (0.53) NPC1TSHR
SCHEMBL15862001 0.73 NPC1 (0.50) NPC1GRM5TSHRKMT2AMAPT
SCHEMBL28568822 0.71 NPC1 (0.52) NPC1GRM5TSHRCYP2C19MAPT
SCHEMBL8116326 0.71 SIGMAR1 (0.48) NPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4482730-A Synthesis of dioxabicyclo[3.2.1]octanes and oxepanes ORTHO PHARMACEUTICAL CORPORATION (US) 1984-11-13 US disclosed
US-4387234-A Synthesis of dioxabicyclo[3.2.1]octanes and oxepanes ORTHO PHARMACEUTICAL CORPORATION (US) 1983-06-07 US disclosed
EP-0012622-B1 1-TOSLOXY-2,2-ETHYLENEDIOXY-6,10-DIMETHYL UNDECANES AND UNDECENES, PROCESS FOR THE PREPARATION OF 2S*,3R*-3-BENZYLOXY-6,6-ETHYLENE DIOXY-2-METHYL-2-(5'-HYDROXY-4'-METHYLPENTYL)-OXEPANE, AND USE OF THE LATTER FOR THE PREPARATION OF OXEPAN-3-OL DERIVATIVES ORTHO PHARMACEUTICAL CORPORATION (US) 1982-12-15 EP disclosed
US-4322353-A Synthesis of dioxabicyclo(3.2.1)octanes and oxepanes ORTHO PHARMACEUTICAL CORPORATION (US) 1982-03-30 US disclosed
EP-0038696-A2 Synthesis of dioxabicyclo(3.2.1.)octanes and oxepanes ORTHO PHARMACEUTICAL CORPORATION (US) 1981-10-28 EP disclosed
US-4256644-A 3-BENZYLOXY-6,6-ETHYLENEDIOXY-2-METHYL-2-(5-HYDROXY-4 -METHYLPENTYL)OXEPANE MADE BY A MULTISTEP PROCESS ORTHO PHARMACEUTICAL CORPORATION (US) 1981-03-17 US disclosed
EP-0012622-A2 1-Tosloxy-2,2-ethylenedioxy-6,10-dimethyl undecanes and undecenes, process for the preparation of 2S*,3R*-3-benzyloxy-6,6-ethylene dioxy-2-methyl-2-(5'-hydroxy-4'-methylpentyl)-oxepane, and use of the latter for the preparation of oxepan-3-ol derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1980-06-25 EP disclosed
US-4188328-A Chemical intermediates in the preparation of oxepane compounds ORTHO PHARMACEUTICAL CORPORATION (US) 1980-02-12 US disclosed