SCHEMBL11048012

SCHEMBL11048012

O=S(=O)(c1ccccc1)c1ncc(Br)cn1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.50
LMNA P02545 3/20 0.44
MAPT P10636 3/20 0.44
HTT P42858 3/20 0.44
ALDH1A1 P00352 5/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
LOXL2 Q9Y4K0 2/20 0.40
AGTR1 P30556 1/20 0.40
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
AURKA O14965 1/20 0.38
FFAR2 O15552 1/20 0.38
KDM4E B2RXH2 1/20 0.37
IDO1 P14902 1/20 0.37
AKR1B1 P15121 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11032457 0.81 GAA (0.54) LMNAMAPTHTTALDH1A1TDP1
SCHEMBL10979591 0.80 HTR6 (0.50) HTR6LMNAMAPTHTTALDH1A1
SCHEMBL10973648 0.80 HTR6 (0.50) HTR6LMNAMAPTHTTALDH1A1
SCHEMBL11063128 0.80 HTR6 (0.50) HTR6LMNAMAPTHTTALDH1A1
SCHEMBL6924070 0.79 HTR6 (0.59) HTR6ALDH1A1HSD17B10TDP1MEN1
SCHEMBL4653156 0.77 AGTR1 (0.57) HTR6LMNAMAPTHTTALDH1A1
SCHEMBL27459397 0.75 HTR6 (0.54) HTR6ALDH1A1HSD17B10TDP1LOXL2
SCHEMBL5610257 0.73 HTR6 (0.52) HTR6ALDH1A1HSD17B10TDP1LOXL2
SCHEMBL8074581 0.73 HTR6 (0.65) HTR6HTTALDH1A1HSD17B10TDP1
SCHEMBL16141 0.72 CA2 (0.48) HTR6LMNAMAPTHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033195-B1 PYRIMIDINE-2-SULPHIDES AND THEIR S-OXIDES FOR USE IN MEDICINE, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, PROCESSES FOR THEIR PREPARATION AND SUCH COMPOUNDS WHEN NOVEL PER SE NYEGAARD & CO. A/S (NO) 1985-12-04 EP disclosed
US-4423047-A INHIBITING ABNORMAL CELL PROLIFERATION NYEGAARD & CO. A/S (NO) 1983-12-27 US disclosed
EP-0033195-A1 Pyrimidine-2-sulphides and their S-oxides for use in medicine, pharmaceutical compositions containing them, processes for their preparation and such compounds when novel per se NYEGAARD & CO. A/S (NO) 1981-08-05 EP disclosed