SCHEMBL11048072

SCHEMBL11048072

c1ccc(CCCCCCC2CCC[N]C2)cc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.44
CYP19A1 P11511 2/20 0.43
SLC18A3 Q16572 1/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
CCR3 P51677 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5250338 1.00 SIGMAR1 (0.44) SIGMAR1CYP19A1SLC18A3OPRM1OPRD1
SCHEMBL8777947 0.98 SIGMAR1 (0.42) SIGMAR1CYP19A1SLC18A3OPRM1OPRD1
SCHEMBL9432698 0.94 SLC18A3 (0.46) SIGMAR1CYP19A1SLC18A3OPRM1OPRD1
SCHEMBL9433185 0.89 CYP19A1 (0.44) SIGMAR1CYP19A1SLC18A3CCR3
SCHEMBL11042566 0.87 CTSS (0.47) OPRM1OPRD1OPRK1
SCHEMBL18435050 0.82 SIGMAR1 (0.61) SIGMAR1CYP19A1SLC18A3OPRM1OPRD1
SCHEMBL8116499 0.81 CYP19A1 (0.47) SIGMAR1CYP19A1SLC18A3CCR3
SCHEMBL8111557 0.81 CYP19A1 (0.47) SIGMAR1CYP19A1SLC18A3CCR3
SCHEMBL7392307 0.80 SIGMAR1 (0.64) SIGMAR1SLC18A3
SCHEMBL5087578 0.80 SIGMAR1 (0.64) SIGMAR1SLC18A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed