SCHEMBL11050032

SCHEMBL11050032

CCC1CNCCC1CC(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A11 P48066 6/20 0.53
SLC6A12 P48065 5/20 0.53
SLC6A13 Q9NSD5 5/20 0.53
SLC6A1 P30531 3/20 0.53
GABRA5 P31644 3/20 0.53
GABRB2 P47870 3/20 0.53
GABRA1 P14867 2/20 0.53
GABRA4 P48169 2/20 0.53
GABRR1 P24046 1/20 0.53
AKR1C4 P17516 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
KCNH2 Q12809 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
TSHR P16473 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11042628 0.98 SLC6A11 (0.52) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5
SCHEMBL11042625 0.84 SLC6A1 (0.39) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5
SCHEMBL11811910 0.82 SLC6A1 (0.42) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5
SCHEMBL11079186 0.81 SLC6A1 (0.37) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5
SCHEMBL11713269 0.81 SLC6A1 (0.37) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5
SCHEMBL11713259 0.81 SLC6A1 (0.37) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5
SCHEMBL11079183 0.81 SLC6A1 (0.37) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5
SCHEMBL11713819 0.80 MAPT (0.38) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5
SCHEMBL11051156 0.80 MAPT (0.38) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5
SCHEMBL11713802 0.80 MAPT (0.38) SLC6A11SLC6A12SLC6A13SLC6A1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4442107-A HYPOTENSIVE, ANTIARRHYTHMIA ACF CHEMIEFARMA N.V. (NL) 1984-04-10 US disclosed
EP-0035821-A1 Quinoline derivatives, pharmaceutical compositions containing such compounds, and method for the preparation of these compounds ACF Chemiefarma N.V. (NL) 1981-09-16 EP disclosed
US-4012396-A Processes and intermediates for cis or trans 2-or 3-(1-acyl-3-vinyl-4-piperidine)acetic or propionic acid esters HOFFMANN-LA ROCHE INC. (US) 1977-03-15 US disclosed
US-3959294-A Processes and intermediates for cis or trans 2- or 3-(1-acyl-3-vinyl-4-piperidine)acetic or propionic acid esters HOFFMANN-LA ROCHE INC. (US) 1976-05-25 US disclosed
US-3957800-A PROCESSES AND INTERMEDIATES FOR CIS OR TRANS 2- OR 3-(1-ACYL-3-VINYL-4-PIPERIDINE)ACETIC OR PROPIONIC ACID ESTERS HOFFMANN-LA ROCHE INC. (US) 1976-05-18 US disclosed