SCHEMBL11050203

SCHEMBL11050203

CCCc1cccc(C)c1-n1cnc(N)nc1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 2/20 0.37
DHFR P00374 2/20 0.36
HSP90AB1 P08238 1/20 0.36
ELANE P08246 2/20 0.34
GRM5 P41594 1/20 0.33
CHRNA7 P36544 1/20 0.33
TLR8 Q9NR97 1/20 0.33
DAO P14920 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
TDP2 O95551 1/20 0.32
ABL1 P00519 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
THRB P10828 1/20 0.32
MPI P34949 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.32
RAB9A P51151 1/20 0.32
DUSP3 P51452 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056242 0.93 HCAR1 (0.40) HCAR1DHFRELANECHRNA7SMN1; SMN2
SCHEMBL11053280 0.92 TLR7 (0.37) HCAR1DHFRCHRNA7TLR8
SCHEMBL11057586 0.92 ELANE (0.36) HCAR1DHFRELANEGRM5TLR8
SCHEMBL11053109 0.91 NPEPPS (0.36) HCAR1DHFRELANEGRM5TLR8
SCHEMBL11052581 0.86 HCAR1 (0.48) HCAR1CHRNA7POLB
SCHEMBL11053171 0.86 ELANE (0.33) HCAR1DHFRELANEGRM5TLR8
SCHEMBL11056344 0.86 EGFR (0.37) HCAR1HSP90AB1ELANECHRNA7KDM4E
SCHEMBL11053265 0.84 HCAR1 (0.38) HCAR1DHFRELANETLR8HTT
SCHEMBL11051199 0.84 ELANE (0.39) DHFRELANEKDM4EPOLBMAPT
SCHEMBL11055480 0.84 APLNR (0.39) DHFRHSP90AB1ELANETLR8SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed