SCHEMBL11052645

SCHEMBL11052645

C#CCNC(=S)N(C(=N)N)c1c(C)cccc1CC

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ALOX12 P18054 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ESR1 P03372 1/20 0.32
ATM Q13315 1/20 0.31
OPRM1 P35372 2/20 0.30
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11051176 0.95 ALDH1A1 (0.32) ALDH1A1ALOX12SMN1; SMN2
SCHEMBL11057623 0.87 ALDH1A1 (0.38) ALDH1A1TP53CYP3A4TDP1SMN1; SMN2
SCHEMBL11053556 0.85 GAA (0.35) ALDH1A1ESR1
SCHEMBL11055264 0.84 ALDH1A1 (0.38) ALDH1A1TP53CYP3A4TDP1ALOX12
SCHEMBL11137837 0.82 ALDH1A1 (0.52) ALDH1A1ALOX12SMN1; SMN2
SCHEMBL11057730 0.82 ALDH1A1 (0.35) ALDH1A1TP53CYP3A4TDP1ALOX12
SCHEMBL11053221 0.81 CA1 (0.34) ALDH1A1TP53CYP3A4TDP1SMN1; SMN2
SCHEMBL11138433 0.81 ALDH1A1 (0.41) ALDH1A1TP53CYP3A4TDP1ALOX12
SCHEMBL11053231 0.81 ALDH1A1 (0.36) ALDH1A1TP53CYP3A4TDP1ALOX12
SCHEMBL11057843 0.79 GAA (0.36) ALDH1A1TP53CYP3A4TDP1ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4418209-A ANTIULCER, ANTIARRYTHMIC, ANTIDIARRHEAL, ANTISPASMODIC, ANTIPARASITIC, AND ANTISECRETORY AGENTS WILLIAM H. RORER, INC. (US) 1983-11-29 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed