SCHEMBL11053231

SCHEMBL11053231

CCc1cccc(C)c1N(C(=N)N)C(=S)NC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
POLB P06746 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALOX12 P18054 1/20 0.33
ESR1 P03372 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
ATM Q13315 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
EGFR P00533 1/20 0.31
MEN1 O00255 1/20 0.30
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11054047 0.87 ALDH1A1 (0.40) ALDH1A1TP53CYP3A4TDP1POLB
SCHEMBL11055264 0.86 ALDH1A1 (0.38) ALDH1A1TP53CYP3A4TDP1SMN1; SMN2
SCHEMBL11138433 0.83 ALDH1A1 (0.41) ALDH1A1TP53CYP3A4TDP1POLB
SCHEMBL11052645 0.81 ALDH1A1 (0.34) ALDH1A1TP53CYP3A4TDP1SMN1; SMN2
SCHEMBL11057843 0.81 GAA (0.36) ALDH1A1TP53CYP3A4TDP1ALOX12
SCHEMBL11060096 0.80 ALDH1A1 (0.36) ALDH1A1TP53CYP3A4TDP1SMN1; SMN2
SCHEMBL11137837 0.80 ALDH1A1 (0.52) ALDH1A1POLBSMN1; SMN2ALOX12TSHR
Hydrochloric Acid SCHEMBL11141378 0.79 GRIN2D (0.35) ALDH1A1TP53CYP3A4TDP1SMN1; SMN2
SCHEMBL11057730 0.79 ALDH1A1 (0.35) ALDH1A1TP53CYP3A4TDP1SMN1; SMN2
SCHEMBL6698678 0.78 TP53 (0.45) ALDH1A1TP53CYP3A4TDP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4418209-A ANTIULCER, ANTIARRYTHMIC, ANTIDIARRHEAL, ANTISPASMODIC, ANTIPARASITIC, AND ANTISECRETORY AGENTS WILLIAM H. RORER, INC. (US) 1983-11-29 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed