SCHEMBL11052878

SCHEMBL11052878

CC(C)(C)NC(=O)NC(=N)Nc1ccc(Br)cc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
ABCB1 P08183 1/20 0.47
ABCC1 P33527 1/20 0.47
RAB9A P51151 5/20 0.46
MAPK1 P28482 4/20 0.46
PKM P14618 2/20 0.46
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
NPC1 O15118 3/20 0.43
ALDH1A1 P00352 2/20 0.42
GLA P06280 1/20 0.42
CASP3 P42574 1/20 0.42
HTT P42858 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
GAA P10253 1/20 0.41
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11057187 0.86 KCNMA1 (0.50) RAB9AMAPK1MEN1KMT2ANPC1
SCHEMBL11055535 0.85 APP (0.54) RAB9AMAPK1PKMMEN1KMT2A
SCHEMBL11053343 0.83 MEN1 (0.60) ABCB1ABCC1RAB9AMAPK1MEN1
SCHEMBL11052503 0.83 KCNMA1 (0.53) RAB9AMAPK1PKMMEN1KMT2A
SCHEMBL11050905 0.83 NPC1 (0.51) KDM4ERAB9AMAPK1MEN1KMT2A
SCHEMBL11579191 0.82 MAPK1 (0.50) KDM4EABCB1ABCC1RAB9AMAPK1
SCHEMBL11055583 0.82 MAPT (0.47) RAB9AMAPK1MEN1KMT2ANPC1
SCHEMBL11579742 0.82 PDK1 (0.53) RAB9AMAPK1MEN1KMT2ANPC1
SCHEMBL11052550 0.82 GAA (0.51) KDM4ERAB9APKMMEN1KMT2A
SCHEMBL11053662 0.81 NPC1 (0.49) KDM4ERAB9AMAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4488993-A Amidinoureas WILLIAM H. RORER, INC. 1984-12-18 US disclosed
US-4220658-A Treatment of hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-02 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed