SCHEMBL11056041

SCHEMBL11056041

O=C(Cc1ccc(Cl)c(Cl)c1)c1ncc[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.48
ALDH1A1 P00352 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
KMT2A Q03164 4/20 0.46
LOXL2 Q9Y4K0 1/20 0.43
MAOB P27338 1/20 0.42
MEN1 O00255 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
CLK1 P49759 1/20 0.41
S1PR5 Q9H228 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
KDM4A O75164 1/20 0.39
KDM5A P29375 1/20 0.39
KDM5B Q9UGL1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981241 0.77 RAB9A (0.41) KMT2ANPC1RAB9A
SCHEMBL6037395 0.76 KMT2A (0.47) KMT2ANPC1RAB9AMAPTSMN1; SMN2
SCHEMBL27702200 0.75 KMT2A (0.40) KMT2AMAOBMEN1
SCHEMBL11485375 0.75 ALDH1A1 (0.47) ALDH1A1KMT2AMEN1NPC1RAB9A
SCHEMBL6432858 0.75 KMT2A (0.46) KMT2ANPC1RAB9AMAPTSMN1; SMN2
SCHEMBL29938476 0.73 KMT2A (0.37) KMT2AMEN1NPC1RAB9ASMN1; SMN2
SCHEMBL10825235 0.72 CYP4F2 (0.38) KMT2ANPC1RAB9AS1PR5
SCHEMBL29938710 0.71 CYP26A1 (0.46) ALDH1A1MAPK1KMT2AMEN1NPC1
SCHEMBL7342304 0.71 BTK (0.39) ALDH1A1MAPK1HSD17B10KMT2AMEN1
SCHEMBL6201848 0.71 S1PR5 (0.58) PIK3CAKMT2AKDM4ES1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4466977-A N-[2-Amino(oxy- or thia- group-substituted-cycloaliphatic)]benzeneacetamides and -benzamide analgesics THE UPJOHN COMPANY (US) 1984-08-21 US disclosed
EP-0108602-A1 N-(2-aminocycloalkyl)benzamide and benzeneacetamide derivatives THE UPJOHN COMPANY (US) 1984-05-16 EP disclosed
US-4360531-A Substituted cycloalkanes THE UPJOHN COMPANY (US) 1982-11-23 US disclosed