SCHEMBL11056042

SCHEMBL11056042

COc1ccc2cc(N(CC(=O)O)C(=O)OC(C)(C)C)ccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 7/20 0.46
AKR1C2 P52895 7/20 0.46
PTGS1 P23219 4/20 0.46
CYP1A2 P05177 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KDM4E B2RXH2 1/20 0.42
KEAP1 Q14145 3/20 0.41
NFE2L2 Q16236 3/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
AKR1C1 Q04828 1/20 0.39
PTGS2 P35354 3/20 0.39
CDC42 P60953 1/20 0.39
RAC1 P63000 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3660817 0.88 KEAP1 (0.49) KEAP1NFE2L2TSHR
SCHEMBL7191809 0.87 ALDH1A1 (0.41) ALDH1A1KDM4EKEAP1NFE2L2
SCHEMBL11052501 0.86 NQO2 (0.39) HSD17B10
SCHEMBL11052784 0.85 MT-CO2 (0.39) CYP1A2ALDH1A1CYP2C19
SCHEMBL8712805 0.84 KDM4E (0.40) AKR1C3AKR1C2PTGS1CYP1A2ALDH1A1
SCHEMBL10978236 0.80 CLK1 (0.44) AKR1C3AKR1C2PTGS1CA2
SCHEMBL28705822 0.79 KDM4E (0.43) AKR1C3AKR1C2PTGS1CYP1A2ALDH1A1
SCHEMBL11649618 0.78 PTPN1 (0.42) HPGDCYP2C19
SCHEMBL8313937 0.77 SMN1; SMN2 (0.40) ALDH1A1
SCHEMBL6715518 0.77 PTGIR (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4490370-A BACTERICIDES ELI LILLY AND COMPANY (US) 1984-12-25 US disclosed
EP-0122155-A2 Improvements in or relating to naphthylglycyl cephalosporin derivatives ELI LILLY AND COMPANY (US) 1984-10-17 EP disclosed