SCHEMBL11056562

SCHEMBL11056562

CCCCCNC(=O)N(C(=N)N)c1c(C)cccc1Br

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 2/20 0.36
ALOX5 P09917 1/20 0.36
HPGD P15428 3/20 0.36
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MGLL Q99685 1/20 0.36
HDAC6 Q9UBN7 2/20 0.35
EPHX1 P07099 3/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
CA2 P00918 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11060199 0.99 NAAA (0.39) NAAAHPGDMAPK1NPSR1L3MBTL1
SCHEMBL11058223 0.96 ALOX5 (0.39) ALOX5HPGDHDAC6ALDH1A1HTT
SCHEMBL11057304 0.92 L3MBTL1 (0.38) ALOX5HPGDMAPK1NPSR1L3MBTL1
Hydrochloric Acid SCHEMBL11556716 0.90 NAAA (0.40) NAAAALOX5HPGDMAPK1NPSR1
Hydrochloric Acid SCHEMBL11561808 0.89 NAAA (0.42) NAAAHPGDMAPK1NPSR1L3MBTL1
Hydrochloric Acid SCHEMBL11561818 0.89 NAAA (0.42) NAAAHPGDMAPK1NPSR1L3MBTL1
Hydrochloric Acid SCHEMBL11558614 0.89 NAAA (0.42) NAAAHPGDMAPK1NPSR1L3MBTL1
Hydrochloric Acid SCHEMBL11565507 0.89 NAAA (0.42) NAAAHPGDMAPK1NPSR1L3MBTL1
SCHEMBL11057738 0.87 TDP1 (0.39) NAAAALOX5HPGDMAPK1NPSR1
Hydrochloric Acid SCHEMBL11562345 0.87 ALOX5 (0.42) NAAAALOX5HPGDALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed