SCHEMBL11056591

SCHEMBL11056591

CCCCCNc1ncn(-c2c(CC)cccc2CC)c(=S)n1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 2/20 0.39
EGFR P00533 1/20 0.37
FGFR1 P11362 1/20 0.37
DNM2 P50570 2/20 0.37
ELANE P08246 2/20 0.36
HRH4 Q9H3N8 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TLR8 Q9NR97 1/20 0.33
MAPK8 P45983 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11050354 0.88 KCNH3 (0.41) KCNH3EGFRFGFR1DNM2ELANE
SCHEMBL11352072 0.86 DNM2 (0.40) KCNH3EGFRFGFR1DNM2ELANE
SCHEMBL11054993 0.86 KCNH2 (0.38) EGFRFGFR1
SCHEMBL11053577 0.84 MKNK1 (0.47) KCNH3
SCHEMBL11053096 0.84 ELANE (0.43) KCNH3EGFRFGFR1ELANEHRH4
SCHEMBL11059128 0.82 KCNH2 (0.37) EGFRFGFR1
SCHEMBL11056312 0.81 LCK (0.44) FGFR1MAPTNPSR1
SCHEMBL11057759 0.81 KCNH3 (0.35) KCNH3
SCHEMBL11053159 0.81 ELANE (0.41) KCNH3EGFRFGFR1DNM2ELANE
SCHEMBL11057771 0.80 FGFR1 (0.46) KCNH3EGFRFGFR1ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed