SCHEMBL11059128

SCHEMBL11059128

CCc1cccc(CC)c1-n1cnc(NC)nc1=S

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.37
SCN5A Q14524 2/20 0.37
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
HCAR1 Q9BXC0 1/20 0.33
KMT2A Q03164 1/20 0.32
EGFR P00533 1/20 0.31
FGFR1 P11362 1/20 0.31
SRC P12931 1/20 0.31
NPEPPS P55786 1/20 0.31
HTR1A P08908 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
CACNA1C Q13936 1/20 0.31
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
GABRA1 P14867 2/20 0.30
GABRB2 P47870 2/20 0.30
PTK2 Q05397 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11054223 0.92 KMT2A (0.36) KCNH2SCN5AALDH1A1HCAR1KMT2A
SCHEMBL11054993 0.87 KCNH2 (0.38) KCNH2SCN5AALDH1A1HPGDKMT2A
SCHEMBL11059651 0.86 HCAR1 (0.44) KCNH2SCN5AALDH1A1LMNAHPGD
SCHEMBL11056006 0.85 KCNH2 (0.39) KCNH2SCN5AALDH1A1LMNAHPGD
SCHEMBL11056595 0.85 CDK4 (0.40) ALDH1A1LMNAHPGDHCAR1KMT2A
SCHEMBL11056217 0.84 ESR1 (0.34) ESR1ESR2
Hydrochloric Acid SCHEMBL11053509 0.84 KCNH2 (0.38) KCNH2SCN5AALDH1A1LMNAHPGD
SCHEMBL11056312 0.83 LCK (0.44) ALDH1A1LMNAKMT2AFGFR1
SCHEMBL11057759 0.83 KCNH3 (0.35) KCNH2SCN5AALDH1A1LMNAHPGD
SCHEMBL11055859 0.83 MKNK1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed