SCHEMBL11057015

SCHEMBL11057015

CCc1cccc(Cl)c1N(C(=N)N)C(=S)NC

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.36
LMNA P02545 3/20 0.33
GAA P10253 3/20 0.33
IDO1 P14902 2/20 0.33
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TAAR1 Q96RJ0 2/20 0.33
KMT2A Q03164 2/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
NR1I2 O75469 1/20 0.32
TP53 P04637 1/20 0.32
CACNA1C Q13936 1/20 0.32
SCN5A Q14524 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
MEN1 O00255 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11060096 0.90 ALDH1A1 (0.36) LMNAGAAHTTSMN1; SMN2TP53
Hydrochloric Acid SCHEMBL11141378 0.89 GRIN2D (0.35) LMNAGAAHTTSMN1; SMN2TP53
Hydrochloric Acid SCHEMBL11137243 0.86 HTT (0.35) PKMLMNAGAAIDO1HTT
SCHEMBL11055264 0.85 ALDH1A1 (0.38) GAAHTTSMN1; SMN2KMT2AEGFR
SCHEMBL10614640 0.85 TP53 (0.35) LMNAGAAIDO1HTTSMN1; SMN2
SCHEMBL11142932 0.84 KMT2A (0.34) PKMGAAHTTSMN1; SMN2KMT2A
SCHEMBL11053970 0.82 GAA (0.39) LMNAGAAHTTSMN1; SMN2KMT2A
Hydrochloric Acid SCHEMBL11141193 0.81 GAA (0.38) LMNAGAAHTTSMN1; SMN2KMT2A
SCHEMBL11053330 0.79 ALDH1A1 (0.35) LMNAIDO1HTTSMN1; SMN2TAAR1
SCHEMBL11057730 0.78 ALDH1A1 (0.35) GAASMN1; SMN2KMT2ATP53CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4418209-A ANTIULCER, ANTIARRYTHMIC, ANTIDIARRHEAL, ANTISPASMODIC, ANTIPARASITIC, AND ANTISECRETORY AGENTS WILLIAM H. RORER, INC. (US) 1983-11-29 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed