SCHEMBL11060096

SCHEMBL11060096

CCc1cccc(CC)c1N(C(=N)N)C(=S)NC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
CACNA1C Q13936 1/20 0.35
SCN5A Q14524 1/20 0.35
GABRA1 P14867 2/20 0.35
GABRB2 P47870 2/20 0.35
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TP53 P04637 2/20 0.33
CYP3A4 P08684 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALOX12 P18054 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GRIN2D O15399 3/20 0.33
GRIN3B O60391 3/20 0.33
GRIN1 Q05586 3/20 0.33
GRIN2A Q12879 3/20 0.33
GRIN2B Q13224 3/20 0.33
GRIN2C Q14957 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11141378 0.98 GRIN2D (0.35) ALDH1A1GAAMAPTCACNA1CSCN5A
SCHEMBL11055264 0.94 ALDH1A1 (0.38) ALDH1A1GAAMAPTCACNA1CSCN5A
SCHEMBL11057015 0.90 PKM (0.36) ALDH1A1GAAMAPTCACNA1CSCN5A
SCHEMBL11142932 0.90 KMT2A (0.34) ALDH1A1GAAMAPTCACNA1CSCN5A
SCHEMBL11057730 0.87 ALDH1A1 (0.35) ALDH1A1GAAMAPTCACNA1CSCN5A
SCHEMBL11059269 0.84 HTT (0.37) ALDH1A1GAAMAPTGABRA1GABRB2
SCHEMBL11141768 0.84 GABRA1 (0.39) ALDH1A1GAAMAPTCACNA1CSCN5A
SCHEMBL11056985 0.84
SCHEMBL11060226 0.84 GRIN2D (0.33) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL11060077 0.83 CACNA1C (0.39) ALDH1A1CACNA1CSCN5AGABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4418209-A ANTIULCER, ANTIARRYTHMIC, ANTIDIARRHEAL, ANTISPASMODIC, ANTIPARASITIC, AND ANTISECRETORY AGENTS WILLIAM H. RORER, INC. (US) 1983-11-29 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed