SCHEMBL11057230

SCHEMBL11057230

CC(C)(C)NC(=O)NC(=N)Nc1ccc(Cl)cc1I

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.43
POLB P06746 2/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39
TRPA1 O75762 1/20 0.39
GRIK1 P39086 1/20 0.38
SERPINE1 P05121 1/20 0.37
PDK1 Q15118 2/20 0.36
PDK2 Q15119 2/20 0.36
PDK3 Q15120 2/20 0.36
PDK4 Q16654 2/20 0.36
ALPL P05186 1/20 0.36
ANO1 Q5XXA6 1/20 0.35
MAPT P10636 1/20 0.35
ATM Q13315 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056102 0.86 HTT (0.36) HTTPOLBKDM4EALDH1A1KMT2A
SCHEMBL11052114 0.86 PDK1 (0.50) HTTPOLBKDM4EALDH1A1KMT2A
SCHEMBL11052830 0.85 POLB (0.58) HTTPOLBKDM4EALDH1A1KMT2A
SCHEMBL11053772 0.85 HTT (0.38) HTTPOLBKMT2AMEN1MAPK1
SCHEMBL11053656 0.85 HTT (0.50) HTTPOLBKDM4EALDH1A1KMT2A
SCHEMBL11053662 0.84 NPC1 (0.49) HTTPOLBKDM4EALDH1A1KMT2A
SCHEMBL11055981 0.84 RAB9A (0.44) HTTPOLBKDM4EALDH1A1KMT2A
SCHEMBL11056677 0.84 HTT (0.46) HTTPOLBKDM4EALDH1A1KMT2A
SCHEMBL11053981 0.84 PDK1 (0.50) HTTPOLBKDM4EALDH1A1KMT2A
SCHEMBL11263600 0.83 GAA (0.48) HTTPOLBALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4488993-A Amidinoureas WILLIAM H. RORER, INC. 1984-12-18 US disclosed
US-4220658-A Treatment of hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-02 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed