SCHEMBL11053772

SCHEMBL11053772

CC(C)(C)NC(=O)NC(=N)Nc1ccc(F)cc1I

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.38
TBXA2R P21731 1/20 0.36
GAA P10253 2/20 0.36
NPC1 O15118 6/20 0.36
RAB9A P51151 6/20 0.36
HDAC1 Q13547 2/20 0.35
PKM P14618 3/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPK1 P28482 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056102 0.88 HTT (0.36) HTTTBXA2RGAANPC1RAB9A
SCHEMBL11054561 0.86 HTT (0.50) HTTGAANPC1RAB9APKM
SCHEMBL11057230 0.85 HTT (0.43) HTTRAB9AMEN1KMT2AMAPK1
SCHEMBL11053662 0.85 NPC1 (0.49) HTTNPC1RAB9AMEN1KMT2A
SCHEMBL11052569 0.85 ALDH1A1 (0.43) HTTTBXA2RNPC1RAB9AMEN1
SCHEMBL11052904 0.84 HTT (0.47) HTTMEN1KMT2AMAPK1POLB
SCHEMBL11052091 0.84 NPC1 (0.40) HTTTBXA2RGAANPC1RAB9A
SCHEMBL11250897 0.84 PKM (0.48) HTTTBXA2RNPC1RAB9APKM
SCHEMBL11053888 0.83 HTT (0.47) HTTNPC1RAB9APKMMEN1
SCHEMBL11050805 0.83 IDH2 (0.39) HTTTBXA2RNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4488993-A Amidinoureas WILLIAM H. RORER, INC. 1984-12-18 US disclosed
US-4220658-A Treatment of hypertension with amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-02 US disclosed
US-4088785-A HYPOTENSIVE AGENTS WILLIAM H. RORER, INC. (US) 1978-05-09 US disclosed