SCHEMBL11057686

SCHEMBL11057686

Cc1cccc(Br)c1-n1cnc(NCCOCc2ccccc2)nc1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
GBA1 P04062 1/20 0.33
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
CHRNA7 P36544 1/20 0.33
HTR1A P08908 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
ABL1 P00519 1/20 0.32
P2RX7 Q99572 1/20 0.32
ALDH1A1 P00352 2/20 0.32
WEE1 P30291 1/20 0.32
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CCND2 P30279 1/20 0.31
CCND3 P30281 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052481 0.91 MKNK1 (0.34) MAOAMAOBMKNK1MKNK2CHRNA7
SCHEMBL11056309 0.89 MEN1 (0.36) MAOAMAOBL3MBTL1GBA1MKNK1
SCHEMBL11059310 0.88 CHRNA7 (0.44) CHRNA7P2RX7
SCHEMBL11053108 0.86 MKNK1 (0.43) MKNK1MKNK2ALDH1A1HTTSMN1; SMN2
SCHEMBL11055490 0.85 MAOA (0.38) MAOAMAOBGBA1MKNK1MKNK2
SCHEMBL11059426 0.80 KMT2A (0.35) MAOAMAOBMKNK1MKNK2CHRNA7
SCHEMBL11053517 0.80 TDP1 (0.38) MAOAMAOBMKNK1MKNK2CHRNA7
SCHEMBL11059003 0.80 FGFR1 (0.39)
SCHEMBL11056733 0.80 ALDH1A1 (0.37) ALDH1A1WEE1CDK4CCND1CCND2
SCHEMBL11055055 0.80 CHRNA7 (0.43) MKNK2CHRNA7P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed