SCHEMBL11057697

SCHEMBL11057697

CCc1cccc(CC)c1-n1cnc(NCc2ccccc2)nc1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.46
FGFR1 P11362 1/20 0.42
KDM4E B2RXH2 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
LMNA P02545 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39
TSHR P16473 1/20 0.39
TMIGD3 P0DMS9 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ATM Q13315 1/20 0.39
CDK1 P06493 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11061665 0.93 KMT2A (0.41) LCKFGFR1KDM4ENPC1MAPT
SCHEMBL11070332 0.89 LCK (0.36) LCKFGFR1KDM4ELMNACASP1
SCHEMBL11056312 0.87 LCK (0.44) LCKFGFR1KDM4ENPC1MAPT
SCHEMBL11056787 0.87 LCK (0.43) LCKFGFR1KDM4ENPC1MAPT
SCHEMBL11051007 0.86 CDK4 (0.42) FGFR1LMNACASP1CASP7HSD17B10
Bromide SCHEMBL11356324 0.85 CDK4 (0.41) FGFR1LMNACASP1CASP7HSD17B10
Hydrochloric Acid SCHEMBL11056068 0.85 CDK4 (0.41) FGFR1LMNACASP1CASP7HSD17B10
SCHEMBL11056400 0.84 EGFR (0.35) FGFR1KDM4ELMNAMKNK1HPGD
SCHEMBL11055490 0.84 MAOA (0.38) LCKTDP1CASP1CASP7HSD17B10
SCHEMBL11059488 0.83 MKNK1 (0.37) CASP1CASP7HSD17B10MKNK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4298608-A LOCAL ANESTHETICS WILLIAM H. RORER, INC. (US) 1981-11-03 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed
US-4198408-A 1,4-DISUBSTITUTED-1,2-DIHYDRO-1,3,5-TRIHZIN-2-ONES WILLIAM H. RORER, INC. (US) 1980-04-15 US disclosed