SCHEMBL11054223

SCHEMBL11054223

CCc1cccc(C)c1-n1cnc(NC)nc1=S

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
HCAR1 Q9BXC0 2/20 0.34
KCNH2 Q12809 1/20 0.34
SCN5A Q14524 1/20 0.34
CHRNA7 P36544 8/20 0.32
ALDH1A1 P00352 1/20 0.32
C5AR1 P21730 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PAK1 Q13153 1/20 0.30
PAK2 Q13177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11059128 0.92 KCNH2 (0.37) KMT2AHCAR1KCNH2SCN5AALDH1A1
SCHEMBL11050195 0.88 HCAR1 (0.39) HCAR1CHRNA7
SCHEMBL11059212 0.87 HCAR1 (0.38) KMT2AMEN1HCAR1KCNH2SCN5A
SCHEMBL11052210 0.86 CDK4 (0.37) KMT2AMEN1HCAR1CHRNA7ALDH1A1
SCHEMBL11056523 0.84 MEN1 (0.33) KMT2AMEN1HCAR1CHRNA7CYP1A2
SCHEMBL11057088 0.84 MEN1 (0.37) KMT2AMEN1
SCHEMBL11057671 0.84 KMT2A (0.42) KMT2AMEN1CHRNA7ALDH1A1
SCHEMBL11057092 0.82 CHRNA7 (0.44) HCAR1CHRNA7
SCHEMBL11056492 0.82 KMT2A (0.37) KMT2AMEN1HCAR1CHRNA7ALDH1A1
SCHEMBL11059651 0.81 HCAR1 (0.44) HCAR1KCNH2SCN5AALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed