SCHEMBL11059487

SCHEMBL11059487

CCc1cccc(C)c1-n1cnc(NCCOCCc2ccccc2)nc1=S

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
MKNK1 Q9BUB5 2/20 0.33
MKNK2 Q9HBH9 2/20 0.33
TMIGD3 P0DMS9 2/20 0.32
ADORA2A P29274 2/20 0.32
ADORA2B P29275 2/20 0.32
ADORA1 P30542 2/20 0.32
CHRNA7 P36544 1/20 0.32
ALDH1A1 P00352 4/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
CYP2C19 P33261 3/20 0.32
USP2 O75604 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
HSD17B10 Q99714 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
TSHR P16473 2/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056376 0.94 MKNK1 (0.36) MEN1KMT2AMKNK1MKNK2TMIGD3
SCHEMBL11059426 0.90 KMT2A (0.35) MEN1KMT2AMKNK1MKNK2TMIGD3
SCHEMBL11060192 0.85 MKNK1 (0.36) MEN1KMT2AMKNK1MKNK2ALDH1A1
SCHEMBL11057671 0.85 KMT2A (0.42) MEN1KMT2ACHRNA7ALDH1A1SMN1; SMN2
SCHEMBL11059488 0.84 MKNK1 (0.37) KMT2AMKNK1MKNK2TMIGD3ADORA2A
SCHEMBL11056309 0.82 MEN1 (0.36) MEN1KMT2AMKNK1MKNK2CHRNA7
SCHEMBL11055055 0.80 CHRNA7 (0.43) MKNK2CHRNA7
SCHEMBL11052481 0.80 MKNK1 (0.34) KMT2AMKNK1MKNK2CHRNA7ALDH1A1
SCHEMBL11053577 0.78 MKNK1 (0.47) MEN1KMT2AMKNK1MKNK2ADORA2A
SCHEMBL11056312 0.78 LCK (0.44) MEN1KMT2AMKNK1TMIGD3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed