SCHEMBL11057671

SCHEMBL11057671

CCc1cccc(C)c1-n1cnc(NCc2ccccc2)nc1=S

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.40
ALDH1A1 P00352 2/20 0.40
ALOX12 P18054 1/20 0.40
LCK P06239 1/20 0.39
LMNA P02545 1/20 0.39
RAD52 P43351 1/20 0.39
ATM Q13315 1/20 0.39
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ELANE P08246 1/20 0.37
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
FGFR1 P11362 1/20 0.36
CHRNA7 P36544 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056312 0.93 LCK (0.44) KMT2AMEN1SMN1; SMN2ALDH1A1LCK
SCHEMBL11057004 0.91 LCK (0.43) SMN1; SMN2ALDH1A1LCKLMNARAD52
SCHEMBL11061665 0.88 KMT2A (0.41) KMT2AMEN1SMN1; SMN2ALDH1A1ALOX12
SCHEMBL11059487 0.85 MEN1 (0.36) KMT2AMEN1SMN1; SMN2ALDH1A1ALOX12
SCHEMBL11054223 0.84 KMT2A (0.36) KMT2AMEN1ALDH1A1CHRNA7
SCHEMBL11056523 0.84 MEN1 (0.33) KMT2AMEN1CHRNA7
SCHEMBL11052210 0.81 CDK4 (0.37) KMT2AMEN1ALDH1A1CHRNA7POLB
SCHEMBL11056787 0.81 LCK (0.43) KMT2AALDH1A1LCKLMNARAB9A
SCHEMBL11057697 0.81 LCK (0.46) SMN1; SMN2LCKLMNAATMRAB9A
SCHEMBL11054993 0.80 KCNH2 (0.38) KMT2AMEN1SMN1; SMN2ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed