SCHEMBL11060192

SCHEMBL11060192

CCc1cccc(CC)c1-n1cnc(NCCOCc2ccccc2)nc1=S

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 4/20 0.36
MKNK2 Q9HBH9 4/20 0.36
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
GBA1 P04062 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
LCK P06239 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CRHR1 P34998 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CCND2 P30279 1/20 0.31
CCND3 P30281 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056376 0.91 MKNK1 (0.36) MKNK1MKNK2SMN1; SMN2LCKALDH1A1
SCHEMBL11055490 0.89 MAOA (0.38) MKNK1MKNK2MAOAMAOBGBA1
SCHEMBL11059487 0.85 MEN1 (0.36) MKNK1MKNK2SMN1; SMN2ALDH1A1MEN1
SCHEMBL11053577 0.85 MKNK1 (0.47) MKNK1MKNK2SMN1; SMN2ALDH1A1MEN1
SCHEMBL11056312 0.84 LCK (0.44) MKNK1SMN1; SMN2LCKALDH1A1MEN1
SCHEMBL11056309 0.84 MEN1 (0.36) MKNK1MKNK2MAOAMAOBGBA1
SCHEMBL11053517 0.83 TDP1 (0.38) MKNK1MKNK2MAOAMAOB
SCHEMBL11059488 0.80 MKNK1 (0.37) MKNK1MKNK2MAOAMAOBSMN1; SMN2
SCHEMBL11497315 0.80 MKNK1 (0.39) MKNK1MKNK2MAOAMAOBSMN1; SMN2
SCHEMBL11054993 0.79 KCNH2 (0.38) SMN1; SMN2ALDH1A1MEN1KMT2ACDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed