SCHEMBL11060153

SCHEMBL11060153

CCc1cccc(CC)c1-n1cnc(N)nc1=S

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
HCAR1 Q9BXC0 1/20 0.34
LMNA P02545 1/20 0.34
MAP3K14 Q99558 1/20 0.34
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
ROCK1 Q13464 1/20 0.33
TLR8 Q9NR97 1/20 0.33
ELANE P08246 1/20 0.33
KMT2A Q03164 1/20 0.33
DHFR P00374 1/20 0.32
NPEPPS P55786 1/20 0.32
GABRA1 P14867 2/20 0.32
GABRB2 P47870 2/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056492 0.92 KMT2A (0.37) ALDH1A1HCAR1MAP3K14TLR8KMT2A
SCHEMBL11053522 0.90 GRM5 (0.36) MAP3K14ROCK1ELANEDHFR
SCHEMBL11053265 0.84 HCAR1 (0.38) ALDH1A1HPGDHCAR1LMNAMAP3K14
SCHEMBL11058224 0.80 HCAR1 (0.41) HCAR1ROCK1KMT2A
SCHEMBL11056509 0.79 GRM1 (0.34) ALDH1A1HPGDHCAR1LMNAKMT2A
SCHEMBL11059128 0.79 KCNH2 (0.37) ALDH1A1HPGDHCAR1LMNAKMT2A
SCHEMBL11053109 0.79 NPEPPS (0.36) ALDH1A1HPGDHCAR1LMNAMAP3K14
SCHEMBL11054993 0.78 KCNH2 (0.38) ALDH1A1HPGDKMT2ANPEPPS
SCHEMBL11057586 0.78 ELANE (0.36) ALDH1A1HPGDHCAR1LMNAMAP3K14
SCHEMBL11056242 0.77 HCAR1 (0.40) HCAR1MAP3K14ELANEKMT2ADHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed