SCHEMBL11061371

SCHEMBL11061371

N#Cc1ccc2cc3c(=O)c(O)ccc-3[nH]c2c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 2/20 0.41
CDK5R1 Q15078 2/20 0.41
ITK Q08881 2/20 0.41
PTPN11 Q06124 1/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
CHEK1 O14757 2/20 0.39
PIN1 Q13526 1/20 0.39
CYP19A1 P11511 1/20 0.38
TDP2 O95551 3/20 0.37
DAO P14920 1/20 0.37
DDO Q99489 1/20 0.37
IMPDH2 P12268 1/20 0.36
IMPDH1 P20839 1/20 0.36
AR P10275 1/20 0.36
CXCR2 P25025 1/20 0.36
FASN P49327 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11616817 0.84 ITK (0.41) CDK5CDK5R1ITKNOS3NOS1
SCHEMBL3735039 0.78 DAO (0.58) CDK5DAO
SCHEMBL3735366 0.76 KDR (0.56) CDK5CDK5R1CHEK1DAODDO
SCHEMBL3396789 0.76 DAO (0.63) NOS3NOS1NOS2PIN1DAO
SCHEMBL11058812 0.75 MEN1 (0.44) CDK5CDK5R1DAODDO
SCHEMBL1080585 0.70 NOS3 (0.51) ITKNOS3NOS1NOS2PIN1
SCHEMBL11056894 0.70 DAO (0.58) CDK5CDK5R1CYP19A1DAO
SCHEMBL10671177 0.69 CYP19A1 (0.61) CDK5CDK5R1ITKCYP19A1IMPDH2
SCHEMBL29651657 0.69 CYP19A1 (0.61) CDK5CDK5R1ITKCYP19A1IMPDH2
SCHEMBL327599 0.67 PIN1 (0.55) NOS3NOS1NOS2PIN1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4474774-A Acridone substituted phosphorus compounds, compositions containing same and insecticidal method of use VELSICOL CHEMICAL CORPORATION (US) 1984-10-02 US disclosed