SCHEMBL11061749

SCHEMBL11061749

CCc1cccc(Cl)c1N(C(=N)N)C(=S)NCCOCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.40
HTT P42858 1/20 0.40
LMNA P02545 2/20 0.36
ACHE P22303 5/20 0.34
NR1I2 O75469 1/20 0.34
ASAH1 Q13510 1/20 0.33
ALDH1A1 P00352 3/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALOX12 P18054 1/20 0.32
MAPK1 P28482 1/20 0.32
PTPN7 P35236 1/20 0.32
DUSP3 P51452 1/20 0.32
PTPN5 P54829 1/20 0.32
PTPN11 Q06124 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11057847 0.93 SMN1; SMN2 (0.41) SMN1; SMN2HTTLMNAACHEASAH1
SCHEMBL11053216 0.89 SMN1; SMN2 (0.43) SMN1; SMN2HTTLMNAACHENR1I2
SCHEMBL11056570 0.84 SMN1; SMN2 (0.37) SMN1; SMN2LMNAACHENR1I2ALDH1A1
SCHEMBL11054620 0.81 SMN1; SMN2 (0.44) SMN1; SMN2HTTLMNANR1I2ASAH1
SCHEMBL11056986 0.80 ALDH1A1 (0.38) SMN1; SMN2LMNAACHEALDH1A1L3MBTL1
SCHEMBL11061902 0.78 SMN1; SMN2 (0.41) SMN1; SMN2HTTLMNAASAH1ALDH1A1
SCHEMBL11056098 0.78 SMN1; SMN2 (0.41) SMN1; SMN2HTTLMNAACHEASAH1
SCHEMBL11057749 0.78 ALDH1A1 (0.46) SMN1; SMN2LMNAALDH1A1MAPTNPSR1
SCHEMBL11057015 0.77 PKM (0.36) SMN1; SMN2HTTLMNANR1I2ALDH1A1
SCHEMBL11054052 0.76 ALDH1A1 (0.50) SMN1; SMN2LMNAALDH1A1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4418209-A ANTIULCER, ANTIARRYTHMIC, ANTIDIARRHEAL, ANTISPASMODIC, ANTIPARASITIC, AND ANTISECRETORY AGENTS WILLIAM H. RORER, INC. (US) 1983-11-29 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed