SCHEMBL11064083

SCHEMBL11064083

CC(C)c1cc(S(C)(=O)=O)[nH]c1C(=O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.48
GABRB1 P18505 1/20 0.48
BCL2 P10415 2/20 0.44
MCL1 Q07820 2/20 0.44
PTGS2 P35354 5/20 0.40
PTGS1 P23219 4/20 0.40
LMNA P02545 3/20 0.40
MAPT P10636 2/20 0.40
CXCR1 P25024 2/20 0.40
CXCR2 P25025 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 2/20 0.40
RECQL P46063 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP3A4 P08684 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
PMP22 Q01453 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11057963 0.81 ALDH1A1 (0.39) PTGS2PTGS1LMNAMAPTCXCR1
SCHEMBL11064057 0.75 GABRA1 (0.49) GABRA1GABRB1BCL2MCL1PTGS2
SCHEMBL11065593 0.73 PTGS2 (0.38) PTGS2LMNAALDH1A1HPGD
SCHEMBL257678 0.69 GABRA1 (0.48) GABRA1GABRB1BCL2MCL1PTGS2
Sulfur Dioxide SCHEMBL11107367 0.66 ALDH1A1 (0.39) PTGS2LMNAALDH1A1CYP3A4HPGD
SCHEMBL1122739 0.66 BCL2 (0.64) GABRA1GABRB1BCL2MCL1PTGS2
SCHEMBL11695892 0.65 BCL2 (0.68) GABRA1GABRB1BCL2MCL1PTGS2
SCHEMBL12648769 0.65 GABRA1 (0.69) GABRA1GABRB1BCL2MCL1PTGS2
SCHEMBL29405385 0.65 GABRA1 (1.00) GABRA1GABRB1BCL2MCL1PTGS2
SCHEMBL10349532 0.65 FABP3 (0.63) GABRA1GABRB1BCL2MCL1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4458081-A ANTIINFLAMMATORY, ANALGESIC, ANTICOAGULANT, MUSCLE RELAXANT SYNTEX (U.S.A.) INC. (US) 1984-07-03 US disclosed
US-4454326-A 5-Aroyl 6-chloro or 6-bromo 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1,1-di-carboxylates SYNTEX (U.S.A.) INC. (US) 1984-06-12 US disclosed
US-4347187-A Process for preparing 5-aroyl 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acids and novel intermediates therein SYNTEX (U.S.A.) INC. (US) 1982-08-31 US disclosed
US-4347186-A Process for preparing 5-aroyl 1,2-dihydro-3-H pyrrolo[1,2-a]pyrrole-1-carboxylic acids and novel intermediates therein SYNTEX (U.S.A.) INC. (US) 1982-08-31 US disclosed