SCHEMBL11065012

SCHEMBL11065012

Brc1ccccc1Cc1cscn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TAAR1 Q96RJ0 3/20 0.41
SLC6A3 Q01959 7/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 1/20 0.40
IDO1 P14902 2/20 0.40
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KDM4E B2RXH2 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
METAP2 P50579 1/20 0.35
METAP1 P53582 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11073422 0.82 SLC6A3 (0.40) MAPTSLC6A3SLC6A2SLC6A4NPC1
SCHEMBL6001756 0.79 SLC6A3 (0.41) TAAR1SLC6A3IDO1NPC1RAB9A
SCHEMBL30839554 0.76 KDM4C (0.40) MAPTSLC6A3KDM4ETSHRMETAP2
SCHEMBL28551226 0.72 L3MBTL1 (0.50) MAPTTAAR1IDO1SMN1; SMN2TDP1
SCHEMBL2093828 0.71 SCN9A (0.47) SLC6A3SLC6A2SLC6A4CYP2D6TDP1
SCHEMBL6286238 0.71 SLC6A3 (0.38) MAPTNPSR1SLC6A3SLC6A2SLC6A4
SCHEMBL8703610 0.71 TAAR1 (0.64) TAAR1IDO1CYP1A2CYP2D6TSHR
SCHEMBL29930048 0.71 TAAR1 (0.64) TAAR1IDO1CYP1A2CYP2D6TSHR
SCHEMBL6287745 0.70 CYP1A2 (0.41) SLC6A3NPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL2793555 0.69 GPR84 (0.59) MAPTTAAR1RAB9AKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4479952-A 1-(4-benzyl-2-thiazolyl) piperazine; antiinflammatory; immunomodulator SCIENCE UNION ET CIE (FR) 1984-10-30 US disclosed